SCHEMBL5522301

SCHEMBL5522301

Cc1cc(C(=O)N[C@H](C(=O)O)c2ccccc2)c(=O)n(Cc2ccc(C(F)(F)F)cc2)c1C

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 4/20 0.47
CNR2 P34972 4/20 0.47
PDE2A O00408 2/20 0.45
PPARG P37231 2/20 0.45
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MTTP P55157 6/20 0.41
KLRK1 P26718 2/20 0.41
MICA Q29983 2/20 0.41
RAET1L Q5VY80 2/20 0.41
S1PR2 O95136 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
TSHR P16473 1/20 0.41
CYP2C19 P33261 1/20 0.41
BRD4 O60885 1/20 0.41
FAAH O00519 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5521539 0.92 PDE2A (0.46) CNR1CNR2PDE2APPARGKDM4E
SCHEMBL27680156 0.92 PDE2A (0.46) CNR1CNR2PDE2APPARGKDM4E
SCHEMBL5522248 0.89 CNR2 (0.50) CNR1CNR2PPARGBRD4FAAH
SCHEMBL2746633 0.89 CNR2 (0.50) CNR1CNR2PPARGBRD4FAAH
SCHEMBL5516376 0.88 KMT2A (0.47) CNR1CNR2PPARGALDH1A1BRD4
SCHEMBL5524739 0.86 ATM (0.52) CNR1CNR2PPARGBRD4FAAH
SCHEMBL5516389 0.83 MEN1 (0.48) CNR1CNR2PPARGALDH1A1BRD4
SCHEMBL5522480 0.81 CNR1 (0.69) CNR1CNR2MTTP
SCHEMBL11922978 0.81 PDE2A (0.43) CNR1CNR2PDE2APPARGKDM4E
SCHEMBL5520940 0.81 CNR2 (0.44) CNR1CNR2PPARGALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8367666-B2 3-carbamoyl-2-pyridone derivatives SHIONOGI & CO., LTD. (JP) 2013-02-05 US disclosed
US-8367666-B2 3-carbamoyl-2-pyridone derivatives SHIONOGI & CO., LTD. (JP) 2013-02-05 US disclosed
US-8178681-B2 methyl 3-methyl-2-{[2-oxo-1-(2-oxo-ethyl)-1,2,5,6,7,8,9,10-octahydro-cycloocta[b]pyridine-3-carbonyl]-amino}-butyrate; cannabinoid receptor agonist; antiinflammatory agent, immunostimulant, analgesic; atopic dermatitis; excellent in photostability, and have excellent transdermal and oral absorbency SHIONOGI & CO., LTD. (JP) 2012-05-15 US disclosed
US-8178681-B2 methyl 3-methyl-2-{[2-oxo-1-(2-oxo-ethyl)-1,2,5,6,7,8,9,10-octahydro-cycloocta[b]pyridine-3-carbonyl]-amino}-butyrate; cannabinoid receptor agonist; antiinflammatory agent, immunostimulant, analgesic; atopic dermatitis; excellent in photostability, and have excellent transdermal and oral absorbency SHIONOGI & CO., LTD. (JP) 2012-05-15 US disclosed