SCHEMBL5524508

SCHEMBL5524508

CCCCn1c(C)c(C)cc(C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c1=O

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 11/20 0.58
ICAM1 P05362 11/20 0.58
ITGAL P20701 11/20 0.58
POLB P06746 2/20 0.56
MAPT P10636 2/20 0.56
HPGD P15428 2/20 0.56
ALDH1A1 P00352 1/20 0.56
CNR1 P21554 1/20 0.55
CNR2 P34972 1/20 0.55
TP53 P04637 1/20 0.54
CCKBR P32239 1/20 0.52
KDM4E B2RXH2 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
ERAP2 Q6P179 1/20 0.52
ALOX15 P16050 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5515093 0.92 KMT2A (0.55) ITGB2ICAM1ITGALPOLBMAPT
SCHEMBL5515967 0.83 CNR2 (0.69) CNR1CNR2
SCHEMBL5517948 0.83 CNR2 (0.69) CNR1CNR2
SCHEMBL2746843 0.83 CNR2 (0.69) CNR1CNR2
SCHEMBL5520544 0.83 CNR1 (0.55) ITGB2ICAM1ITGALPOLBMAPT
SCHEMBL15780958 0.78 ITGB2 (0.79) ITGB2ICAM1ITGALPOLBMAPT
SCHEMBL5522035 0.78 CNR2 (0.59) CNR1CNR2
SCHEMBL5524532 0.78 CNR2 (0.58) CNR1CNR2
SCHEMBL5524556 0.76 CNR2 (0.57) POLBALDH1A1CNR1CNR2KDM4E
SCHEMBL21001416 0.76 MEN1 (0.66) ITGB2ICAM1ITGALPOLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8367666-B2 3-carbamoyl-2-pyridone derivatives SHIONOGI & CO., LTD. (JP) 2013-02-05 US disclosed
US-8367666-B2 3-carbamoyl-2-pyridone derivatives SHIONOGI & CO., LTD. (JP) 2013-02-05 US disclosed
US-8178681-B2 methyl 3-methyl-2-{[2-oxo-1-(2-oxo-ethyl)-1,2,5,6,7,8,9,10-octahydro-cycloocta[b]pyridine-3-carbonyl]-amino}-butyrate; cannabinoid receptor agonist; antiinflammatory agent, immunostimulant, analgesic; atopic dermatitis; excellent in photostability, and have excellent transdermal and oral absorbency SHIONOGI & CO., LTD. (JP) 2012-05-15 US disclosed
US-8178681-B2 methyl 3-methyl-2-{[2-oxo-1-(2-oxo-ethyl)-1,2,5,6,7,8,9,10-octahydro-cycloocta[b]pyridine-3-carbonyl]-amino}-butyrate; cannabinoid receptor agonist; antiinflammatory agent, immunostimulant, analgesic; atopic dermatitis; excellent in photostability, and have excellent transdermal and oral absorbency SHIONOGI & CO., LTD. (JP) 2012-05-15 US disclosed