SCHEMBL5528216

SCHEMBL5528216

O=c1[nH]ccc2nc(-c3ccc(CNCc4ccc(S)cc4)cc3)c(-c3ccccc3)cc12

nearest known ligand 0.54

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.54
AKT1 P31749 18/20 0.49
AKT2 P31751 6/20 0.48
KCNH2 Q12809 4/20 0.46
HRH2 P25021 1/20 0.42
ADRA1A P35348 1/20 0.42
ADRA1B P35368 1/20 0.42
SLC6A3 Q01959 1/20 0.42
AKT3 Q9Y243 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2893852 0.90 JAK2 (0.55) JAK2AKT1AKT2KCNH2HRH2
SCHEMBL2898847 0.89 JAK2 (0.54) JAK2AKT1AKT2KCNH2
SCHEMBL2890607 0.88 JAK2 (0.53) JAK2AKT1AKT2KCNH2HRH2
SCHEMBL2893767 0.87 JAK2 (0.52) JAK2AKT1AKT2KCNH2
SCHEMBL2893868 0.87 AKT1 (0.53) JAK2AKT1AKT2KCNH2HRH2
SCHEMBL2897765 0.87 JAK2 (0.52) JAK2AKT1AKT2KCNH2
SCHEMBL2893676 0.87 JAK2 (0.52) JAK2AKT1AKT2KCNH2HRH2
SCHEMBL2896812 0.86 JAK2 (0.51) JAK2AKT1AKT2KCNH2
SCHEMBL2890730 0.86 JAK2 (0.51) JAK2AKT1AKT2KCNH2
SCHEMBL2890411 0.85 JAK2 (0.50) JAK2AKT1AKT2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1737861-A1 INHIBITORS OF AKT ACTIVITY Merck & Co., Inc. (US) 2007-01-03 EP claimed
WO-2005100356-A1 INHIBITORS OF AKT ACTIVITY MERCK & CO., INC. (US) 2005-10-27 WO claimed