SCHEMBL5529862

SCHEMBL5529862

CNc1nc(N)nc2cc(-c3c(N4CCCC4)cccc3C(F)(F)F)ccc12.CNc1nc(N)nc2cc(-c3c(SC)cccc3C(F)(F)F)ccc12

nearest known ligand 0.63

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 14/20 0.63
HRH4 Q9H3N8 2/20 0.37
TRPV1 Q8NER1 2/20 0.33
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 1/20 0.32
RECQL P46063 1/20 0.32
NLRP3 Q96P20 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4527626 0.93 PTPN1 (0.68) PTPN1HRH4TRPV1CYP1A2CYP2D6
SCHEMBL4535077 0.89 PTPN1 (0.67) PTPN1HRH4CYP1A2CYP2D6CYP2C19
SCHEMBL4523209 0.81 PTPN1 (0.67) PTPN1HRH4NLRP3
SCHEMBL4527944 0.80 PTPN1 (0.57) PTPN1HRH4TRPV1CYP1A2CYP2D6
SCHEMBL4529240 0.79 PTPN1 (0.53) PTPN1HRH4NLRP3
SCHEMBL4531449 0.79 PTPN1 (0.53) PTPN1CYP1A2CYP2D6CYP2C19RECQL
Trifluoroacetic Acid SCHEMBL4522538 0.78 PTPN1 (0.58) PTPN1HRH4
SCHEMBL13040908 0.77 PTPN1 (1.00) PTPN1
SCHEMBL4532451 0.77 PTPN1 (0.51) PTPN1TRPV1NLRP3
SCHEMBL3732057 0.77 PTPN1 (1.00) PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1812409-A1 AMINOQUINAZOLINES COMPOUNDS F. Hoffmann-Roche AG (CH) 2007-08-01 EP disclosed
WO-2006050843-A1 AMINOQUINAZOLINES COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2006-05-18 WO disclosed