SCHEMBL5534906

SCHEMBL5534906

CC1CN(c2ccc(C3CN(c4nc(-c5ccncc5F)cc(=O)n4C)CCO3)cc2)CC(C)N1

nearest known ligand 0.79

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 18/20 0.79
CYP2D6 P10635 12/20 0.79
CYP1A2 P05177 8/20 0.79
CSNK1A1 P48729 1/20 0.57
GSK3A P49840 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL81558 1.00 GSK3B (0.79) GSK3BCYP2D6CYP1A2CSNK1A1GSK3A
SCHEMBL88164 0.91 GSK3B (0.80) GSK3BCYP2D6CYP1A2CSNK1A1GSK3A
SCHEMBL87674 0.91 GSK3B (0.85) GSK3BCYP2D6CYP1A2CSNK1A1GSK3A
SCHEMBL84001 0.90 GSK3B (0.81) GSK3BCYP2D6CYP1A2CSNK1A1GSK3A
SCHEMBL88183 0.90 GSK3B (0.84) GSK3BCYP2D6CYP1A2CSNK1A1GSK3A
SCHEMBL87722 0.90 GSK3B (0.84) GSK3BCYP2D6CYP1A2CSNK1A1GSK3A
SCHEMBL88433 0.89 GSK3B (0.82) GSK3BCYP2D6CYP1A2CSNK1A1GSK3A
SCHEMBL82880 0.89 GSK3B (0.82) GSK3BCYP2D6CYP1A2CSNK1A1GSK3A
SCHEMBL87770 0.89 GSK3B (0.81) GSK3BCYP2D6CYP1A2CSNK1A1GSK3A
SCHEMBL88036 0.88 GSK3B (1.00) GSK3BCYP2D6CYP1A2CSNK1A1GSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1805164-A2 6-(PYRIDINYL)-4-PYRIMIDONE DERIVATES AS TAU PROTEIN KINASE 1 INHIBITORS Mitsubishi Pharma Corporation (JP) 2007-07-11 EP claimed
WO-2006036015-A2 6- (PYRIDINYL) -4-PYRIMIDONE DERIVATES AS TAU PROTEIN KINASE 1 INHIBITORS MITSUBISHI PHARMA CORPORATION (JP) 2006-04-06 WO claimed