SCHEMBL5543919

SCHEMBL5543919

Cn1c(CN2CCC[C@H]3CCc4cccnc4[C@H]32)nc2cccc(N3CC[N+](C(=O)[O-])(C(C)(C)C)CC3)c21

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 5/20 0.44
CYP2D6 P10635 1/20 0.44
OPRL1 P41146 1/20 0.32
KCNH2 Q12809 1/20 0.32
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
FNTA P49354 5/20 0.31
FNTB P49356 5/20 0.31
CHRM5 P08912 2/20 0.30
CHRM1 P11229 2/20 0.30
EGLN1 Q9GZT9 1/20 0.30
CHRM2 P08172 1/20 0.30
CHRM4 P08173 1/20 0.30
CHRM3 P20309 1/20 0.30
MAPT P10636 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4166416 0.85 CXCR4 (0.59) CXCR4CYP2D6KCNH2
SCHEMBL4177280 0.84 CXCR4 (0.47) CXCR4CYP2D6FNTAFNTB
SCHEMBL4181823 0.84 CXCR4 (0.53) CXCR4CYP2D6KCNH2CHRM5CHRM1
SCHEMBL13875189 0.72 CXCR4 (0.41) CXCR4CYP2D6FNTAFNTB
SCHEMBL4185850 0.72 CXCR4 (0.41) CXCR4CYP2D6FNTAFNTB
SCHEMBL4171448 0.72 CXCR4 (0.41) CXCR4CYP2D6FNTAFNTB
SCHEMBL4171449 0.72 CXCR4 (0.41) CXCR4CYP2D6FNTAFNTB
SCHEMBL4179325 0.71 CXCR4 (0.51) CXCR4CYP2D6KCNH2FNTAFNTB
SCHEMBL13875218 0.71 CXCR4 (0.51) CXCR4CYP2D6KCNH2FNTAFNTB
SCHEMBL4173707 0.71 CXCR4 (0.51) CXCR4CYP2D6KCNH2FNTAFNTB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1853604-A2 CHEMICAL COMPOUNDS SmithKline Beecham Corporation (US) 2007-11-14 EP disclosed
WO-2006096444-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-09-14 WO disclosed