SCHEMBL5552201

SCHEMBL5552201

Cc1cc2c([nH]1)CCN(C(=O)c1ccc(CNC(=O)OC(C)(C)C)c(C)c1)c1ccccc1-2

nearest known ligand 0.53

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 18/20 0.53
PDCD1 Q15116 2/20 0.47
CD274 Q9NZQ7 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5552241 0.85 AVPR2 (0.53) AVPR2PDCD1CD274
Hydrochloric Acid SCHEMBL5552018 0.81 PDCD1 (0.47) AVPR2PDCD1CD274
SCHEMBL5552618 0.81 AVPR2 (0.46) AVPR2PDCD1CD274
SCHEMBL2130987 0.80 AVPR2 (0.51) AVPR2PDCD1CD274
SCHEMBL5232067 0.70 AVPR2 (0.66) AVPR2
SCHEMBL5231560 0.70 AVPR2 (0.66) AVPR2
SCHEMBL2705385 0.69 AVPR2 (0.42) AVPR2PDCD1CD274
SCHEMBL6627507 0.69 AVPR2 (1.00) AVPR2
SCHEMBL1495979 0.69 EPHX2 (0.64) AVPR2
SCHEMBL18917226 0.69 AVPR2 (0.42) AVPR2PDCD1CD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781661-A2 VASOPRESSIN V1A ANTAGONISTS Ferring B.V. (NL) 2007-05-09 EP disclosed
WO-2006021213-A2 VASOPRESSIN V1A ANTAGONISTS FERRING B.V. (NL) 2006-03-02 WO disclosed