SCHEMBL5552246

SCHEMBL5552246

Cc1cc(C(=O)N2Cc3cnn(C)c3Nc3ccccc32)ccc1CCC(=O)N1CCC(CN(Cc2ccccc2)C2CCNCC2)CC1

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 18/20 0.54
OXTR P30559 11/20 0.52
AVPR2 P30518 6/20 0.52
CHRM2 P08172 1/20 0.49
CHRM4 P08173 1/20 0.49
CHRM5 P08912 1/20 0.49
CHRM3 P20309 1/20 0.49
DRD3 P35462 1/20 0.49
OPRK1 P41145 1/20 0.49
TSPO P30536 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2864446 0.90 AVPR1A (0.57) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL2865882 0.88 AVPR1A (0.55) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL2131724 0.86 AVPR1A (0.64) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL2131897 0.85 AVPR1A (0.67) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL2866241 0.85 AVPR1A (0.64) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL2863935 0.84 AVPR1A (0.60) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL2129977 0.84 AVPR1A (0.59) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL2129672 0.84 AVPR1A (0.65) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL2858555 0.84 AVPR1A (0.60) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL2128795 0.83 AVPR1A (0.62) AVPR1AOXTRAVPR2CHRM2CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781661-A2 VASOPRESSIN V1A ANTAGONISTS Ferring B.V. (NL) 2007-05-09 EP claimed
WO-2006021213-A2 VASOPRESSIN V1A ANTAGONISTS FERRING B.V. (NL) 2006-03-02 WO claimed