SCHEMBL5553972

SCHEMBL5553972

CCC(C(=O)Oc1ccc2c(c1F)c(CC(=O)O)c(C)n2C(=O)c1ccc(F)c(F)c1)c1c(C)n(C(=O)c2ccc(F)c(F)c2)c2ccc(O)c(F)c12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 8/20 0.39
AKR1C2 P52895 8/20 0.39
PTGS1 P23219 3/20 0.38
PTGS2 P35354 3/20 0.38
AKR1C4 P17516 2/20 0.36
AKR1C1 Q04828 2/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
PTGES O14684 1/20 0.36
ABCC3 O15438 1/20 0.36
ABCC4 O15439 1/20 0.36
ABCB11 O95342 1/20 0.36
MT-CO2 P00403 1/20 0.36
LMNA P02545 1/20 0.36
ALB P02768 1/20 0.36
CYP1A2 P05177 1/20 0.36
ABCB1 P08183 1/20 0.36
ALOX5 P09917 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
CXCL8 P10145 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5801077 0.91 AKR1C3 (0.47) AKR1C3AKR1C2PTGS1PTGS2AKR1C4
SCHEMBL5560517 0.91 AKR1C3 (0.40) AKR1C3AKR1C2PTGS1PTGS2AKR1C4
SCHEMBL5800728 0.86 AKR1C3 (0.37) AKR1C3AKR1C2PTGS1PTGS2AKR1C4
SCHEMBL5798800 0.85 AKR1C3 (0.39) AKR1C3AKR1C2PTGS1PTGS2AKR1C4
SCHEMBL5796494 0.84 AKR1C3 (0.40) AKR1C3AKR1C2PTGS1PTGS2AKR1C4
SCHEMBL5554232 0.84 AKR1C3 (0.52) AKR1C3AKR1C2PTGS1PTGS2AKR1C4
SCHEMBL6425563 0.82 AKR1C3 (0.35) AKR1C3AKR1C2PTGS1PTGS2MEN1
SCHEMBL6425839 0.82 AKR1C3 (0.35) AKR1C3AKR1C2PTGS1PTGS2MEN1
SCHEMBL5801188 0.82 AKR1C3 (0.39) AKR1C3AKR1C2PTGS1PTGS2AKR1C4
SCHEMBL5797204 0.81 AKR1C3 (0.38) AKR1C3AKR1C2PTGS1PTGS2AKR1C4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1643961-A4 COX-2 AND FAAH INHIBITORS MICROBIA INC (US) 2007-09-12 EP disclosed
EP-1643961-A2 COX-2 AND FAAH INHIBITORS Microbia, Inc. (US) 2006-04-12 EP disclosed
WO-2005002525-A2 COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2005-01-13 WO disclosed