SCHEMBL5560580

SCHEMBL5560580

CN(CC=N)NC(=O)c1c[nH]c(=O)c(F)c1Nc1ccc(Br)cc1F

nearest known ligand 0.45

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 20/20 0.45
MAP2K2 P36507 3/20 0.42
ABCB11 O95342 1/20 0.37
NQO2 P16083 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5178279 0.81 MAP2K1 (0.61) MAP2K1MAP2K2ABCB11NQO2
SCHEMBL5559992 0.80 MAP2K1 (0.52) MAP2K1MAP2K2ABCB11NQO2
SCHEMBL5554511 0.79 MAP2K1 (0.53) MAP2K1MAP2K2ABCB11NQO2
SCHEMBL5555084 0.79 MAP2K1 (0.52) MAP2K1MAP2K2ABCB11NQO2
SCHEMBL3455907 0.78 MAP2K1 (0.51) MAP2K1MAP2K2ABCB11NQO2
SCHEMBL5560204 0.78 MAP2K1 (0.66) MAP2K1MAP2K2ABCB11NQO2
SCHEMBL388574 0.78 MAP2K1 (0.61) MAP2K1MAP2K2
SCHEMBL388765 0.77 MAP2K1 (0.53) MAP2K1MAP2K2ABCB11NQO2
SCHEMBL5559526 0.76 MAP2K1 (0.60) MAP2K1MAP2K2ABCB11NQO2
SCHEMBL5560829 0.76 MAP2K1 (0.52) MAP2K1MAP2K2ABCB11NQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1682138-A4 HETEROCYCLIC INHIBITORS OF MEK AND METHODS OF USE THEREOF ARRAY BIOPHARMA INC (US) 2007-01-24 EP disclosed
EP-1682138-A2 HETEROCYCLIC INHIBITORS OF MEK AND METHODS OF USE THEREOF Array Biopharma, Inc. (US) 2006-07-26 EP disclosed
WO-2005051301-A2 HETEROCYCLIC INHIBITORS OF MEK AND METHODS OF USE THEREOF ARRAY BIOPHARMA INC. (US) 2005-06-09 WO disclosed