SCHEMBL5564043

SCHEMBL5564043

Cc1cc2c(cc1Cl)NC(=O)CC(c1cccc(-c3cc(C)[n+]([O-])c(C)c3)c1)=N2

nearest known ligand 0.61

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 4/20 0.61
CYP3A4 P08684 4/20 0.56
GRM3 Q14832 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5557357 0.94 GRM2 (0.69) GRM2CYP3A4GRM3
SCHEMBL5562802 0.86 GRM2 (0.73) GRM2CYP3A4GRM3
SCHEMBL6486875 0.85 CYP3A4 (0.77) GRM2CYP3A4GRM3
SCHEMBL5557541 0.84 CYP3A4 (0.73) GRM2CYP3A4GRM3
SCHEMBL5564545 0.83 GRM2 (0.63) GRM2CYP3A4GRM3
SCHEMBL5557849 0.82 CYP3A4 (0.74) GRM2CYP3A4GRM3
SCHEMBL5557774 0.82 GRM2 (0.88) GRM2CYP3A4GRM3
SCHEMBL5563357 0.82 GRM2 (0.67) GRM2CYP3A4GRM3
SCHEMBL5562130 0.82 GRM2 (0.67) GRM2CYP3A4GRM3
SCHEMBL5556725 0.80 GRM2 (0.71) GRM2CYP3A4GRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1474416-B1 DIHYDROBENZODIAZEPIN-2-ONE-DERIVATIVES FOR THE TREATMENT OF NEUROLOGICAL DISORDERS HOFFMANN LA ROCHE (CH) 2007-09-26 EP disclosed