SCHEMBL5570845

SCHEMBL5570845

[CH2]c1ccc2c(c1)CN(C)CC2c1cc2ccccc2o1

nearest known ligand 0.76

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 18/20 0.76
SLC6A4 P31645 18/20 0.76
SLC6A3 Q01959 17/20 0.76
CYP2D6 P10635 1/20 0.45
KCNH2 Q12809 1/20 0.45
CHRNB2 P17787 1/20 0.41
CHRNA4 P43681 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4302124 0.87 SLC6A2 (0.77) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL4302131 0.86 SLC6A2 (1.00) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL4308536 0.86 SLC6A2 (0.76) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL4317608 0.86 SLC6A2 (0.76) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL4313447 0.84 SLC6A4 (0.72) SLC6A2SLC6A4SLC6A3
SCHEMBL4455109 0.83 SLC6A4 (0.71) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL4301931 0.83 SLC6A4 (0.71) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL4317129 0.83 SLC6A2 (0.71) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL4307020 0.82 SLC6A2 (0.69) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL4456866 0.82 SLC6A2 (0.69) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1778639-A2 ARYL-AND HETEROARYL-SUBSTITUTED TETRAHYDROISOQUINOLINES AND USE THEREOF TO BLOCK REUPTAKE OF NOREPINEPHRINE, DOPAMINE, AND SEROTONIN AMR Technology, Inc. (US) 2007-05-02 EP disclosed
WO-2006020049-A2 ARYL-AND HETEROARYL-SUBSTITUTED TETRAHYDROISOQUINOLINES AND USE THEREOF TO BLOCK REUPTAKE OF NOREPINEPHRINE, DOPAMINE, AND SEROTONIN AMR TECHNOLOGY, INC. (US) 2006-02-23 WO disclosed