SCHEMBL5574152

SCHEMBL5574152

CCC(c1ccc(Nc2nccc3ccncc23)cc1)[C@H](NC1=C(SC(C)C)C(=O)C12CCCCC2)C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 4/20 0.42
ITGA4 P13612 4/20 0.42
MEN1 O00255 1/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
KMT2A Q03164 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3836320 0.93 ITGB1 (0.36) ITGB1ITGA4
SCHEMBL3833596 0.90 MEN1 (0.32) ITGB1ITGA4MEN1NPC1RAB9A
SCHEMBL3833845 0.89 ITGB1 (0.38) ITGB1ITGA4
SCHEMBL3833793 0.88 ITGB1 (0.38) ITGB1ITGA4
SCHEMBL3836800 0.86 ITGB1 (0.34) ITGB1ITGA4
SCHEMBL3832798 0.86 ITGB1 (0.38) ITGB1ITGA4
SCHEMBL6131672 0.86 ITGB1 (0.38) ITGB1ITGA4
SCHEMBL3884133 0.85 ITGB1 (0.58) ITGB1ITGA4
SCHEMBL2978337 0.85 ITGB1 (0.58) ITGB1ITGA4
SCHEMBL3836404 0.82 ITGB1 (0.42) ITGB1ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1780201-A2 PHENYLALANINE ENAMIDE DERIVATIVES POSSESSING A CYCLOBUTENE GROUP, FOR USE AS INTEGRIN INHIBITORS Celltech R&D Limited (GB) 2007-05-02 EP disclosed