SCHEMBL5574241

SCHEMBL5574241

CC1(C)C(=O)C=C1NC(Cc1ccc(Oc2nccc3ccncc23)cc1)C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 11/20 0.51
ITGA4 P13612 11/20 0.51
PPARG P37231 6/20 0.37
FFAR1 O14842 1/20 0.36
DRD1 P21728 1/20 0.36
GPR132 Q9UNW8 1/20 0.35
PPARA Q07869 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2982542 1.00 ITGB1 (0.51) ITGB1ITGA4PPARGFFAR1DRD1
SCHEMBL5147510 0.91 ITGB1 (0.44) ITGB1ITGA4FFAR1DRD1
SCHEMBL2978167 0.89 ITGB1 (0.45) ITGB1ITGA4PPARGFFAR1DRD1
SCHEMBL2978173 0.89 ITGB1 (0.45) ITGB1ITGA4PPARGFFAR1DRD1
SCHEMBL2978120 0.89 ITGB1 (0.42) ITGB1ITGA4PPARGFFAR1DRD1
SCHEMBL2974021 0.86 ITGB1 (0.54) ITGB1ITGA4PPARG
SCHEMBL7265369 0.86 ITGB1 (0.54) ITGB1ITGA4PPARG
SCHEMBL2980127 0.84 ITGB1 (0.53) ITGB1ITGA4
SCHEMBL5147594 0.83 PPARG (0.44) ITGB1ITGA4PPARGFFAR1DRD1
SCHEMBL5147512 0.82 FFAR1 (0.38) ITGB1ITGA4FFAR1DRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1780201-A2 PHENYLALANINE ENAMIDE DERIVATIVES POSSESSING A CYCLOBUTENE GROUP, FOR USE AS INTEGRIN INHIBITORS Celltech R&D Limited (GB) 2007-05-02 EP disclosed