SCHEMBL5579211

SCHEMBL5579211

O=c1cc(-c2ccccn2)oc2ccccc12

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 1/20 0.68
CYP1B1 Q16678 3/20 0.63
CYP1A1 P04798 2/20 0.63
CYP1A2 P05177 2/20 0.63
TNKS O95271 6/20 0.58
NPC1 O15118 4/20 0.58
GABRP O00591 4/20 0.58
GABRD O14764 4/20 0.58
GABRA1 P14867 4/20 0.58
GABRB1 P18505 4/20 0.58
GABRG2 P18507 4/20 0.58
GABRB3 P28472 4/20 0.58
GABRA5 P31644 4/20 0.58
GABRA3 P34903 4/20 0.58
GABRA2 P47869 4/20 0.58
GABRB2 P47870 4/20 0.58
GABRA4 P48169 4/20 0.58
GABRE P78334 4/20 0.58
GABRA6 Q16445 4/20 0.58
GABRG1 Q8N1C3 4/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30307539 1.00 AHR (0.68) AHRCYP1B1CYP1A1CYP1A2TNKS
SCHEMBL11558273 0.81 TNKS (0.53) AHRCYP1B1CYP1A1CYP1A2TNKS
SCHEMBL11561361 0.81 AHR (0.56) AHRCYP1B1CYP1A1CYP1A2TNKS
SCHEMBL312714 0.79 TNKS (0.62) CYP1B1CYP1A2TNKSNPC1GABRP
SCHEMBL4174237 0.79 AHR (0.61) AHRCYP1B1CYP1A1CYP1A2TNKS
SCHEMBL4183286 0.79 AHR (0.61) AHRCYP1B1CYP1A1CYP1A2TNKS
SCHEMBL12278333 0.78 AHR (0.56) AHRCYP1B1CYP1A1CYP1A2NPC1
SCHEMBL4181907 0.78 AHR (0.53) AHRCYP1B1CYP1A1CYP1A2PLA2G2A
SCHEMBL1868748 0.77 GRM4 (0.65) AHRCYP1B1TNKSNPC1GABRP
Flavone SCHEMBL28996632 0.77 TNKS (0.70) CYP1B1CYP1A2TNKSNPC1GABRP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070148185-A1 Novel therapeutic target for protozoal diseases VIRGINIA POLYTECHNIC INSTITUTE AND STATE UNIVERSITY 2007-06-28 US disclosed
EP-0388188-B1 Benzoxepin derivatives SUNTORY LTD (JP) 1994-01-12 EP disclosed
US-5041444-A Hypoglycemic agents; anticoagulants SUNTORY LIMITED (JP) 1991-08-20 US disclosed
EP-0388188-A1 Benzoxepin derivatives SUNTORY LIMITED (JP) 1990-09-19 EP disclosed