SCHEMBL5580152

SCHEMBL5580152

CCC(Cc1ccc(Cl)cc1)(NC(=O)c1cccc2ccccc12)C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 3/20 0.49
ACP3 P15309 1/20 0.48
PLK1 P53350 1/20 0.44
NR1H4 Q96RI1 1/20 0.44
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
ALDH1A1 P00352 2/20 0.42
HPGD P15428 2/20 0.42
HSP90AA1 P07900 1/20 0.42
MAPT P10636 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
RAB9A P51151 1/20 0.42
HDAC8 Q9BY41 2/20 0.42
MMP3 P08254 1/20 0.42
ANO1 Q5XXA6 1/20 0.41
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC2 Q92769 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5580154 1.00 DRD4 (0.49) DRD4ACP3PLK1NR1H4MEN1
SCHEMBL5580180 0.90 DEGS1 (0.49) DRD4PLK1NR1H4MEN1KMT2A
SCHEMBL5580183 0.90 DEGS1 (0.49) DRD4PLK1NR1H4MEN1KMT2A
SCHEMBL5580159 0.85 CCR3 (0.49) MEN1KMT2AMAPT
SCHEMBL5580161 0.85 CCR3 (0.49) MEN1KMT2AMAPT
SCHEMBL5580151 0.76 CCR3 (0.49) NR1H4MEN1KMT2AALDH1A1MAPT
SCHEMBL5580149 0.76 CCR3 (0.49) NR1H4MEN1KMT2AALDH1A1MAPT
SCHEMBL5580405 0.75 APEX1 (0.44) KMT2AALDH1A1MAPT
SCHEMBL5580402 0.75 APEX1 (0.44) KMT2AALDH1A1MAPT
SCHEMBL485144 0.73 CXCR2 (0.56) MEN1KMT2AALDH1A1HPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6420424-B1 ADMINISTERING PHENYLALANINE AMIDE DERIVATIVES (SUCH AS S-ETHYL-2-AMINO-3-(4-CHLOROPHENYL)PROPIONATE HYDROCHLORIDE) TO TREAT ALLERGIC DISORDERS, INCLUDING ASTHMA, RHINITIS, DERMATITUS, AND PRURITIS SMITHKLINE BEECHAM CORPORATION 2002-07-16 US claimed
US-20070249915-A1 Inhibitors SHISEIDO COMPANY, LTD. (JP) 2007-10-25 US disclosed