SCHEMBL5582513

SCHEMBL5582513

CCc1cccc(CNCC(C([AsH2])Cc2cc(F)cc(F)c2)[C@H](Sc2nnc3nc(C)cc(C)n23)C(=O)O)c1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.41
ALDH1A1 P00352 5/20 0.39
BACE1 P56817 7/20 0.38
CTSD P07339 2/20 0.38
KDM4E B2RXH2 4/20 0.37
POLB P06746 1/20 0.36
CTSB P07858 4/20 0.35
HPGD P15428 2/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C19 P33261 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5582515 1.00 MAPK1 (0.41) MAPK1ALDH1A1BACE1CTSDKDM4E
SCHEMBL5582514 1.00 MAPK1 (0.41) MAPK1ALDH1A1BACE1CTSDKDM4E
SCHEMBL5579871 0.91 MAPK1 (0.41) MAPK1ALDH1A1BACE1CTSDKDM4E
SCHEMBL5579867 0.91 MAPK1 (0.41) MAPK1ALDH1A1BACE1CTSDKDM4E
SCHEMBL5579876 0.91 MAPK1 (0.41) MAPK1ALDH1A1BACE1CTSDKDM4E
SCHEMBL5127703 0.82 MAPK1 (0.37) MAPK1ALDH1A1BACE1CTSDKDM4E
SCHEMBL5127700 0.77 MAPK1 (0.36) MAPK1ALDH1A1BACE1CTSDKDM4E
SCHEMBL3348528 0.77 BACE1 (0.49) ALDH1A1BACE1CTSDKDM4EPOLB
SCHEMBL3348521 0.77 BACE1 (0.49) ALDH1A1BACE1CTSDKDM4EPOLB
SCHEMBL5131022 0.71 BACE1 (0.39) ALDH1A1BACE1CTSDCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7294642-B2 1,3-Diamino-2-hydroxypropane pro-drug derivatives ELAN PHARMACEUTICALS, INC. (US) 2007-11-13 US disclosed