SCHEMBL5591968

SCHEMBL5591968

CC(OCC1(c2ccccc2)CCN(C)CC1)c1cc(C#N)ccc1-c1cccc(C(F)(F)F)c1

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 14/20 0.55
SLC6A4 P31645 8/20 0.47
KCNH2 Q12809 5/20 0.47
TACR3 P29371 1/20 0.41
MCHR1 Q99705 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5592183 0.90 TACR1 (0.53) TACR1
SCHEMBL5591972 0.82 TACR1 (0.60) TACR1SLC6A4KCNH2
SCHEMBL3590174 0.81 TACR1 (0.71) TACR1SLC6A4KCNH2TACR3
SCHEMBL3587308 0.81 TACR1 (0.71) TACR1SLC6A4KCNH2TACR3
SCHEMBL12050245 0.78 TACR1 (0.60) TACR1SLC6A4KCNH2TACR3
SCHEMBL5591980 0.78 TACR1 (0.45) TACR1SLC6A4KCNH2
SCHEMBL2424007 0.73 TACR1 (0.51) TACR1SLC6A4KCNH2TACR3
SCHEMBL3603008 0.73 TACR1 (0.59) TACR1TACR3
SCHEMBL13962479 0.73 TACR1 (0.49) TACR1SLC6A4KCNH2
SCHEMBL3586496 0.71 TACR1 (0.67) TACR1TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007121389-A2 4,4-DISUBSTITUTED PIPERIDINE DERIVATIVES AS NK-I AND SEROTONIN TRANSPORTER INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-10-25 WO disclosed