SCHEMBL5591981

SCHEMBL5591981

N#Cc1ccc(-c2ccccc2)c(CCOCC2(c3ccccc3)CCNCC2)c1

nearest known ligand 0.51

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 10/20 0.50
SLC6A4 P31645 2/20 0.43
KCNH2 Q12809 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5592184 0.89 TACR1 (0.58) TACR1SLC6A4
SCHEMBL5592059 0.81 TACR1 (0.53) TACR1SLC6A4
SCHEMBL5591972 0.77 TACR1 (0.60) TACR1SLC6A4KCNH2
SCHEMBL5591980 0.76 TACR1 (0.45) TACR1SLC6A4KCNH2
SCHEMBL5592010 0.76 TACR1 (0.64) TACR1
SCHEMBL5592203 0.73 TACR1 (0.83) TACR1
SCHEMBL1388730 0.73 TACR1 (0.77) TACR1SLC6A4KCNH2
SCHEMBL1388510 0.73 TACR1 (0.71) TACR1SLC6A4KCNH2
Hydrochloric Acid SCHEMBL8114845 0.72 TACR1 (0.75) TACR1SLC6A4KCNH2
SCHEMBL8123020 0.72 TACR1 (0.58) TACR1SLC6A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007121389-A2 4,4-DISUBSTITUTED PIPERIDINE DERIVATIVES AS NK-I AND SEROTONIN TRANSPORTER INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-10-25 WO disclosed