SCHEMBL5592244

SCHEMBL5592244

N#Cc1ccc(-c2cc(Cl)cc(CCOCC3(c4ccccc4)CCN(C(=O)O)CC3)c2)cc1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 4/20 0.49
MCHR1 Q99705 7/20 0.41
CYP3A4 P08684 2/20 0.40
TSHR P16473 2/20 0.40
USP2 O75604 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HTR1A P08908 1/20 0.38
DRD4 P21917 1/20 0.38
HTR2A P28223 1/20 0.38
HRH1 P35367 1/20 0.38
OPRM1 P35372 1/20 0.38
ALDH1A1 P00352 1/20 0.37
CYP2C9 P11712 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3597398 0.91 TACR1 (0.59) TACR1
SCHEMBL5592007 0.90 TACR1 (0.51) TACR1MCHR1CYP3A4TSHRUSP2
SCHEMBL5591983 0.87 TACR1 (0.67) TACR1
SCHEMBL3599074 0.83 TACR1 (0.62) TACR1
SCHEMBL13404451 0.81 TACR1 (0.61) TACR1
SCHEMBL3597348 0.80 TACR1 (0.59) TACR1
SCHEMBL3585726 0.80 TACR1 (0.62) TACR1
SCHEMBL3591749 0.80 TACR1 (0.59) TACR1
SCHEMBL3595413 0.80 TACR1 (0.45) TACR1MCHR1
SCHEMBL3597281 0.77 TACR1 (0.57) TACR1MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007121389-A2 4,4-DISUBSTITUTED PIPERIDINE DERIVATIVES AS NK-I AND SEROTONIN TRANSPORTER INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-10-25 WO disclosed