SCHEMBL5593503

SCHEMBL5593503

COc1cc(F)c(-c2c(OC)nc3ncnn3c2NC(C)C(F)(F)F)cc1F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.38
GRM8 O00222 1/20 0.36
GRM7 Q14831 1/20 0.36
GRM4 Q14833 1/20 0.36
ABL1 P00519 1/20 0.34
EGFR P00533 1/20 0.34
HCK P08631 1/20 0.34
SRC P12931 1/20 0.34
KDR P35968 1/20 0.34
PIK3CB P42338 1/20 0.34
MTOR P42345 1/20 0.34
PIK3CG P48736 1/20 0.34
EPHB4 P54760 1/20 0.34
PRKDC P78527 1/20 0.34
PI4KB Q9UBF8 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.32
HPGD P15428 2/20 0.32
MAPK1 P28482 2/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5593105 0.92 CYP1A2 (0.36) CYP1A2GRM8GRM7GRM4ABL1
SCHEMBL5593334 0.90 MAPK1 (0.34) CYP1A2ABL1SMN1; SMN2MAPK1KDM4E
SCHEMBL5593188 0.90 CYP1A2 (0.42) CYP1A2GRM8GRM7GRM4ABL1
SCHEMBL5593077 0.88 CYP1A2 (0.35) CYP1A2GRM8GRM7GRM4ABL1
SCHEMBL5593152 0.87 CYP1A2 (0.36) CYP1A2GRM8GRM7GRM4ABL1
SCHEMBL5593068 0.86 GRM8 (0.36) CYP1A2GRM8GRM7GRM4ABL1
SCHEMBL5593367 0.83 SMN1; SMN2 (0.36) CYP1A2GRM8GRM7GRM4ABL1
SCHEMBL5593340 0.83 CYP1A2 (0.39) CYP1A2GRM8GRM7GRM4SMN1; SMN2
SCHEMBL5593039 0.82 CYP1A2 (0.40) CYP1A2GRM8GRM7GRM4ABL1
SCHEMBL5593399 0.82 MAPK1 (0.34) CYP1A2SMN1; SMN2HPGDMAPK1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007099092-A1 SUBSTITUTED 6-PHENYL-7-AMINO[1,2,4]-TRIAZOLO[1,5-a]PYRIMIDINES AND THEIR USE FOR CONTROLLING PATHOGENIC FUNGI BASF SE (DE) 2007-09-07 WO claimed