SCHEMBL5594865

SCHEMBL5594865

N#Cc1ccc(NC(=O)Nc2ccccc2-c2ccccc2)c(O)c1.N#Cc1ccc(NC(=O)Nc2ccccc2-c2ccccc2)c(O)c1

nearest known ligand 0.71

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 7/20 0.71
CXCR1 P25024 3/20 0.71
CA12 O43570 2/20 0.48
CA1 P00915 2/20 0.48
CA2 P00918 2/20 0.48
CA9 Q16790 2/20 0.48
RET P07949 1/20 0.46
FLT1 P17948 1/20 0.46
KDR P35968 1/20 0.46
MAPK14 Q16539 1/20 0.46
ALDH1A1 P00352 2/20 0.44
NTRK1 P04629 2/20 0.44
PTGDR2 Q9Y5Y4 1/20 0.43
KDM4E B2RXH2 1/20 0.43
GAA P10253 1/20 0.43
MEN1 O00255 1/20 0.43
CYP2C9 P11712 1/20 0.43
HPGD P15428 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3709514 1.00 CXCR2 (0.71) CXCR2CXCR1CA12CA1CA2
SCHEMBL5595077 0.84 CXCR2 (0.85) CXCR2CXCR1CA12CA1CA2
SCHEMBL7489930 0.83 CXCR2 (1.00) CXCR2CXCR1CA12CA1CA2
SCHEMBL7514963 0.82 CXCR2 (0.73) CXCR2CXCR1CA12CA1CA2
SCHEMBL6824309 0.81 CXCR2 (1.00) CXCR2CXCR1ALDH1A1GAAMEN1
SCHEMBL3705632 0.81 CXCR2 (1.00) CXCR2CXCR1ALDH1A1GAAMEN1
SCHEMBL3710548 0.81 CXCR2 (0.71) CXCR2CXCR1CA12CA1CA2
SCHEMBL7493701 0.80 STAT3 (0.51) CXCR2CXCR1CA12CA1CA2
SCHEMBL27576146 0.80 CXCR2 (0.69) CXCR2CA12CA1CA2CA9
SCHEMBL7489080 0.79 CXCR2 (0.67) CXCR2CXCR1ALDH1A1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0809492-A4 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2007-01-24 EP disclosed
EP-0809492-A1 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-12-03 EP disclosed
WO-1996025157-A1 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1996-08-22 WO disclosed