SCHEMBL5599236

SCHEMBL5599236

CCOC(=O)c1cc(C#N)c(N2CC3CN(C(=O)OC(C)(C)C)CC3C2)nc1C.Cc1nc(N2CC3CN(C(=O)NS(=O)(=O)c4ccccc4)CC3C2)c(C#N)cc1C(=O)O

nearest known ligand 0.84

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
P2RY12 Q9H244 20/20 0.84
CHRM2 P08172 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2C9 P11712 1/20 0.52
DRD3 P35462 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4097633 0.91 P2RY12 (1.00) P2RY12CHRM2CYP3A4CYP2C9DRD3
SCHEMBL4098256 0.85 P2RY12 (0.63) P2RY12CYP3A4CYP2C9
SCHEMBL4098057 0.81 P2RY12 (1.00) P2RY12CHRM2CYP3A4CYP2C9DRD3
SCHEMBL4104695 0.80 P2RY12 (1.00) P2RY12CHRM2CYP3A4CYP2C9DRD3
SCHEMBL5599233 0.79 P2RY12 (0.62) P2RY12
SCHEMBL4105389 0.79 P2RY12 (0.94) P2RY12CHRM2CYP3A4CYP2C9DRD3
SCHEMBL4105011 0.79 P2RY12 (0.79) P2RY12CHRM2CYP3A4CYP2C9DRD3
SCHEMBL4109623 0.79 P2RY12 (1.00) P2RY12CHRM2CYP3A4CYP2C9DRD3
SCHEMBL4105040 0.77 P2RY12 (0.79) P2RY12CHRM2CYP3A4CYP2C9DRD3
SCHEMBL4097854 0.77 P2RY12 (1.00) P2RY12CHRM2CYP3A4CYP2C9DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006073361-A9 NOVEL PYRIDINE COMPOUNDS ASTRAZENECA AB (SE) 2007-08-02 WO disclosed