SCHEMBL5608090

SCHEMBL5608090

CN(C)[N]S(=O)(=O)c1cccc2ccccc12

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 6/20 0.56
F2 P00734 5/20 0.56
PRSS2 P07478 5/20 0.56
PRSS3 P35030 5/20 0.56
CA2 P00918 2/20 0.52
CA1 P00915 1/20 0.52
CA9 Q16790 1/20 0.52
HTR2A P28223 1/20 0.46
HTR2C P28335 1/20 0.46
HTR6 P50406 2/20 0.44
HCRTR1 O43613 1/20 0.43
C1R P00736 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
TSHR P16473 2/20 0.42
SIGMAR1 Q99720 1/20 0.41
KEAP1 Q14145 1/20 0.40
NFE2L2 Q16236 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5610254 0.79 F2 (0.61) PRSS1F2PRSS2PRSS3CA2
SCHEMBL6580084 0.79 F2 (0.65) PRSS1F2PRSS2PRSS3CA2
SCHEMBL9840763 0.77 F2 (0.68) PRSS1F2PRSS2PRSS3CA2
SCHEMBL3248145 0.76 CA1 (0.57) PRSS1F2PRSS2PRSS3CA2
SCHEMBL18537467 0.76 CA1 (0.57) PRSS1F2PRSS2PRSS3CA2
SCHEMBL10652362 0.75 F2 (0.56) PRSS1F2PRSS2PRSS3CA2
SCHEMBL2878187 0.75 F2 (0.56) PRSS1F2PRSS2PRSS3CA2
Trimethylammonium SCHEMBL23581573 0.74 CA1 (0.55) PRSS1F2PRSS2PRSS3CA2
Trimethylammonium SCHEMBL29177484 0.74 CA1 (0.55) PRSS1F2PRSS2PRSS3CA2
Hydrochloric Acid SCHEMBL28348315 0.74 HTR2A (0.55) PRSS1F2PRSS2PRSS3CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1846380-A1 CARDIOVASCULAR COMPOUNDS COMPRISING HETEROCYCLIC NITRIC OXIDE DONOR GROUP COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2007-10-24 EP disclosed
WO-2006078995-A1 CARDIOVASCULAR COMPOUNDS COMPRISING HETEROCYCLIC NITRIC OXIDE DONOR GROUP COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2006-07-27 WO disclosed
WO-2002014261-A2 4-SUBSTITUTED D-GLUTAMIC ACID DERIVATIVES FOR USE AS ANTIBIOTIC ELI LILLY AND COMPANY (US) 2002-02-21 WO disclosed