SCHEMBL5608097

SCHEMBL5608097

CC(=O)c1ccc(Nc2cccc(C)c2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 3/20 0.62
AKR1C2 P52895 3/20 0.62
NPSR1 Q6W5P4 1/20 0.61
ALDH1A1 P00352 3/20 0.57
MAPT P10636 3/20 0.57
HPGD P15428 2/20 0.57
HSD17B10 Q99714 1/20 0.56
RAB9A P51151 7/20 0.53
NPC1 O15118 6/20 0.53
KMT2A Q03164 4/20 0.51
MEN1 O00255 3/20 0.51
RXFP1 Q9HBX9 1/20 0.51
TP53 P04637 1/20 0.51
SMN1; SMN2 Q16637 5/20 0.51
KDM4E B2RXH2 2/20 0.51
TAAR1 Q96RJ0 1/20 0.50
GAA P10253 1/20 0.50
LMNA P02545 2/20 0.49
HTT P42858 1/20 0.49
POLB P06746 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9186732 0.86 AKR1C3 (0.58) AKR1C3AKR1C2NPSR1ALDH1A1MAPT
SCHEMBL5455532 0.86 NPSR1 (0.67) AKR1C3AKR1C2NPSR1ALDH1A1MAPT
SCHEMBL4113285 0.83 NPC1 (0.74) ALDH1A1MAPTHPGDHSD17B10RAB9A
SCHEMBL10523964 0.83 NPSR1 (0.86) NPSR1ALDH1A1MAPTHPGDHSD17B10
SCHEMBL30145137 0.83 NPSR1 (0.86) NPSR1ALDH1A1MAPTHPGDHSD17B10
SCHEMBL1922070 0.83 NPSR1 (0.86) NPSR1ALDH1A1MAPTHPGDHSD17B10
SCHEMBL9071956 0.82 AKR1C3 (0.69) AKR1C3AKR1C2NPSR1ALDH1A1MAPT
SCHEMBL5460527 0.81 AKR1C3 (0.67) AKR1C3AKR1C2ALDH1A1MAPTHPGD
SCHEMBL5608717 0.81 MAPT (0.61) AKR1C3AKR1C2ALDH1A1MAPTHPGD
SCHEMBL9478869 0.81 MAPT (0.71) AKR1C3AKR1C2ALDH1A1MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1354887-B1 Ligands for metals and improved metal-catalyzed processes based thereon MASSACHUSETTS INST TECHNOLOGY (US) 2007-04-25 EP disclosed
EP-1097158-B1 LIGANDS FOR METALS AND METAL-CATALYZED PROCESSES MASSACHUSETTS INST TECHNOLOGY (US) 2006-01-25 EP disclosed
EP-1354887-A1 Ligands for metals and improved metal-catalyzed processes based thereon Massachusetts Insitute of Technology (US) 2003-10-22 EP disclosed
EP-1097158-A2 LIGANDS FOR METALS AND METAL-CATALYZED PROCESSES MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2001-05-09 EP disclosed
WO-2000002887-A2 LIGANDS FOR METALS AND METAL-CATALYZED PROCESSES MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2000-01-20 WO disclosed