SCHEMBL5608592

SCHEMBL5608592

NC(=O)c1ccc(-c2cccc(C(N)=O)c2-c2nccs2)c(C(N)=O)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 1/20 0.46
MYC P01106 1/20 0.39
CTSA P10619 1/20 0.38
TYK2 P29597 1/20 0.37
HDAC2 Q92769 2/20 0.37
KEAP1 Q14145 1/20 0.37
NFE2L2 Q16236 1/20 0.37
SIRT2 Q8IXJ6 1/20 0.37
SIRT1 Q96EB6 1/20 0.37
SIRT3 Q9NTG7 1/20 0.37
CSNK1A1 P48729 1/20 0.36
TYRO3 Q06418 1/20 0.36
DYRK1B Q9Y463 1/20 0.36
F2 P00734 1/20 0.36
F10 P00742 1/20 0.36
PLG P00747 1/20 0.36
F7 P08709 1/20 0.36
F3 P13726 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC4 P56524 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30810276 0.81 PARP1 (0.45) CHEK2MYCTYK2HDAC2KEAP1
SCHEMBL5609015 0.78 CHEK2 (0.43) CHEK2MYCCTSAHDAC2KAT6A
SCHEMBL3201031 0.77 PARP1 (0.46) CTSAKEAP1NFE2L2PARP1
SCHEMBL27664694 0.76 CHEK2 (0.53) CHEK2MYCCTSATYK2HDAC2
SCHEMBL30810193 0.76 HPGD (0.42) CHEK2MYCTYK2SIRT3ADORA2A
SCHEMBL3201989 0.75 CTSA (0.45) CTSAPARP1
SCHEMBL28031696 0.75 SMN1; SMN2 (0.42) CHEK2TYK2PARP1
SCHEMBL3147427 0.75 ADORA2A (0.42) CHEK2TYK2HDAC2KEAP1NFE2L2
SCHEMBL918767 0.74 CSNK1A1 (0.48) CHEK2TYK2HDAC2KEAP1NFE2L2
SCHEMBL2303493 0.74 KAT6A (0.55) CHEK2MYCHDAC2SIRT2SIRT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1805132-A2 NOVEL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2007-07-11 EP disclosed
WO-2006110173-A2 NOVEL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-10-19 WO disclosed