SCHEMBL5613872

SCHEMBL5613872

O=C(O)Cc1cccc(OCC(Oc2cccc(C(O)(C(F)(F)F)C(F)(F)F)c2)c2ccccc2)c1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NR1H3 Q13133 11/20 0.47
NR1H2 P55055 9/20 0.47
PPARG P37231 1/20 0.42
PPARA Q07869 1/20 0.42
MEN1 O00255 1/20 0.42
NR1I2 O75469 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
RXRA P19793 1/20 0.42
VHL P40337 1/20 0.42
RECQL P46063 1/20 0.42
BLM P54132 1/20 0.42
KMT2A Q03164 1/20 0.42
SLC6A9 P48067 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3980467 1.00 NR1H3 (0.47) NR1H3NR1H2PPARGPPARAMEN1
SCHEMBL3977202 0.93 NR1H3 (0.53) NR1H3NR1H2PPARGPPARARXRA
SCHEMBL3977176 0.90 NR1H3 (0.51) NR1H3NR1H2PPARGPPARAMEN1
SCHEMBL3977208 0.89 CACNA1B (0.46) NR1H3NR1H2ALDH1A1SLC6A9
SCHEMBL3975906 0.83 NR1H2 (0.56) NR1H3NR1H2PPARGMEN1KMT2A
SCHEMBL3984317 0.81 NR1H3 (0.47) NR1H3NR1H2PPARGPPARAMEN1
SCHEMBL10680256 0.76 CYP1A2 (0.56) NR1H3NR1H2MEN1MAPTRXRA
SCHEMBL3981981 0.75 PLA2G4B (0.53) NR1H3NR1H2PPARGPPARAMEN1
SCHEMBL3981070 0.74 NR1H3 (0.41) NR1H3NR1H2MEN1KMT2ASLC6A9
SCHEMBL3976637 0.73 MRGPRX4 (0.56)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1802566-A1 HEXAFLUOROISOPROPANOL SUBSTITUTED ETHER DERIVATIVES F. Hoffmann-Roche AG (CH) 2007-07-04 EP claimed
WO-2006037480-A1 HEXAFLUOROISOPROPANOL SUBSTITUTED ETHER DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2006-04-13 WO claimed