SCHEMBL5616660

SCHEMBL5616660

COc1ccc2c(c1Cl)C[C@]1(CCOc3ccccc3)CCC(=O)C=C21

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 8/20 0.41
ESR1 P03372 5/20 0.41
MEN1 O00255 4/20 0.35
KMT2A Q03164 4/20 0.35
ALDH1A1 P00352 3/20 0.35
GAA P10253 1/20 0.35
POLB P06746 1/20 0.33
P4HB P07237 1/20 0.33
NR3C1 P04150 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4782328 0.83 ESR2 (0.45) ESR2ESR1ALDH1A1NR3C1
SCHEMBL4732373 0.83 ESR2 (0.45) ESR2ESR1ALDH1A1NR3C1
SCHEMBL5460555 0.83 ESR2 (0.45) ESR2ESR1ALDH1A1NR3C1
SCHEMBL2421182 0.82 ESR2 (0.58) ESR2ESR1
SCHEMBL2415516 0.71 ESR2 (0.60) ESR2ESR1
SCHEMBL5612544 0.67 CYP19A1 (0.40)
SCHEMBL5616667 0.64 KDM4E (0.40) ALDH1A1GAA
SCHEMBL2420989 0.64 ESR2 (0.58) ESR2ESR1
SCHEMBL2419019 0.63 ESR2 (0.59) ESR2ESR1
SCHEMBL1658799 0.62 ESR2 (0.50) ESR2ESR1MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007081895-A2 PREPARATION OF SUBSTITUTED 2-HYDROXYGIBBA-1(10A), 2, 4, 4B-TETRAEN-6-ONES MERCK & CO., INC. (US) 2007-07-19 WO disclosed