SCHEMBL5620530

SCHEMBL5620530

CCCN1CCCCC1c1nc2c(C(N)=O)cccc2n1CCN1CCCCC1CC

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 14/20 0.57
PARP2 Q9UGN5 4/20 0.43
THRB P10828 1/20 0.40
HTR1A P08908 3/20 0.38
TERT O14746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7705473 0.99 PARP1 (0.56) PARP1PARP2THRBHTR1A
SCHEMBL5619904 0.89 PARP1 (0.67) PARP1PARP2THRBTERT
SCHEMBL5622515 0.88 PARP1 (0.61) PARP1PARP2THRB
SCHEMBL5621717 0.87 PARP1 (0.60) PARP1PARP2
SCHEMBL5621375 0.86 PARP1 (0.57) PARP1PARP2
SCHEMBL7041326 0.86 PARP1 (0.43) PARP1THRBTERT
SCHEMBL5620956 0.86 PARP1 (0.57) PARP1PARP2HTR1A
SCHEMBL5621063 0.86 PARP1 (0.57) PARP1PARP2HTR1A
SCHEMBL5620500 0.86 PARP1 (0.59) PARP1PARP2HTR1A
SCHEMBL5621352 0.85 PARP1 (0.52) PARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39608-E1 Substituted benzimidazoles and their use as PARP inhibitors ABBOTT GMBH & CO. KG (DE) 2007-05-01 US disclosed