SCHEMBL5628142

SCHEMBL5628142

CN1CCN(C(=O)c2ccc3n2Cc2ccc(C(=O)O)cc2N(C(=O)c2ccc(C4CCCCC4)cc2)C3)CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 3/20 0.41
SLC6A7 Q99884 1/20 0.39
MYC P01106 2/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
RAD52 P43351 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
BMPR1B O00238 1/20 0.36
BMPR1A P36894 1/20 0.36
TGFBR1 P36897 1/20 0.36
ACVRL1 P37023 1/20 0.36
ACVR1 Q04771 1/20 0.36
HTR2B P41595 1/20 0.35
MGLL Q99685 2/20 0.35
AVPR1A P37288 1/20 0.35
KMO O15229 1/20 0.35
HSD11B1 P28845 1/20 0.35
POLB P06746 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5626384 0.91 HPGD (0.41) AVPR2SLC6A7ALDH1A1LMNARAD52
Hydrochloric Acid SCHEMBL5628265 0.90 HPGD (0.42) AVPR2SLC6A7ALDH1A1LMNARAD52
SCHEMBL5628972 0.88 AVPR2 (0.48) AVPR2SLC6A7ALDH1A1LMNARAD52
SCHEMBL5629638 0.86 AVPR2 (0.46) AVPR2SLC6A7ALDH1A1LMNARAD52
SCHEMBL5626957 0.80 AVPR1A (0.42) AVPR2SLC6A7ALDH1A1LMNAHTR2B
SCHEMBL5627644 0.79 NAMPT (0.44) AVPR2SLC6A7ALDH1A1LMNARAD52
SCHEMBL5626780 0.79 TSHR (0.45) AVPR2SLC6A7HTR2BMGLLAVPR1A
SCHEMBL5626594 0.78 AVPR1A (0.47) AVPR2SLC6A7ALDH1A1LMNARAD52
SCHEMBL5626277 0.78 AVPR1A (0.48) AVPR2SLC6A7ALDH1A1HTR2BAVPR1A
SCHEMBL5626387 0.78 EPHX2 (0.42) AVPR2SLC6A7ALDH1A1LMNARAD52

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7202239-B2 Cyclohexylphenyl carboxamides tocolytic oxytocin receptor antagonists WYETH (US) 2007-04-10 US claimed
US-7202239-B2 Cyclohexylphenyl carboxamides tocolytic oxytocin receptor antagonists WYETH (US) 2007-04-10 US disclosed
EP-1377582-A1 NOVEL 3-C(O)R SUBSTITUTED 10-CYCLOHEXYLBENZOYL PYRROLOBENZODIAZEPINES; TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS Wyeth (US) 2004-01-07 EP disclosed
WO-2002085907-A1 NOVEL 3-C(O)R SUBSTITUTED 10-CYCLOHEXYLBENZOYL PYRROLOBENZODIAZEPINES; TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS WYETH (US) 2002-10-31 WO disclosed