SCHEMBL5633233

SCHEMBL5633233

Oc1c(Br)cc(CNCC2CCN(CCCCCC(c3ccc(F)cc3)c3ccc(F)cc3)C2)cc1Br

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 14/20 0.76
SCN5A Q14524 1/20 0.41
FAAH O00519 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
TSHR P16473 1/20 0.40
ALOX12 P18054 1/20 0.40
MAPK1 P28482 1/20 0.40
MTOR P42345 1/20 0.40
RAB9A P51151 1/20 0.40
CACNA1F O60840 1/20 0.40
HTR1A P08908 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
DRD4 P21917 1/20 0.40
DRD5 P21918 1/20 0.40
HRH2 P25021 1/20 0.40
ADRA1D P25100 1/20 0.40
HTR2A P28223 1/20 0.40
HTR7 P34969 1/20 0.40
ADRA1A P35348 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5634945 0.86 KCNH2 (1.00) KCNH2
SCHEMBL14476192 0.85 KCNH2 (0.73) KCNH2SCN5ACYP3A4CYP2D6ADORA3
SCHEMBL5633732 0.84 KCNH2 (1.00) KCNH2
SCHEMBL5635444 0.83 KCNH2 (1.00) KCNH2
SCHEMBL5633525 0.81 KCNH2 (0.82) KCNH2
SCHEMBL5024699 0.79 KCNH2 (0.72) KCNH2SCN5AFAAHCYP3A4CYP2D6
SCHEMBL5633170 0.72 KCNH2 (1.00) KCNH2
SCHEMBL5634775 0.72 KCNH2 (1.00) KCNH2
SCHEMBL5633239 0.70 KCNH2 (0.42) KCNH2FAAHCYP3A4CYP2D6TSHR
SCHEMBL5634420 0.70 KCNH2 (1.00) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7244758-B2 N-type calcium channel blockers NEUROMED PHARMACEUTICALS LTD. (CA) 2007-07-17 US claimed
US-20050014748-A1 N-type calcium channel blockers NEUROMED TECHNOLOGIES INC. 2005-01-20 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050014748-A1 N-type calcium channel blockers CACNA1B, CACNA1C, CACNA1I KCNH2 33/4885SCN5A 74/4885FAAH 946/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.