SCHEMBL5633347

SCHEMBL5633347

CCCCN(Cc1ccc(C(N)=O)c(CC(=O)O)c1)Cc1c(-c2ccc(OC)cc2)nc(-c2ccccc2)n1CCCC

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
C5AR1 P21730 1/20 0.40
PTGDR2 Q9Y5Y4 2/20 0.37
TSPO P30536 2/20 0.37
GNRHR P30968 1/20 0.36
MAPT P10636 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
CNR2 P34972 1/20 0.35
NR1H3 Q13133 2/20 0.35
PPARG P37231 3/20 0.35
PPARA Q07869 2/20 0.35
HDAC1 Q13547 1/20 0.35
PARP1 P09874 2/20 0.35
ATP4A P20648 1/20 0.34
ATP4B P51164 1/20 0.34
LTB4R2 Q9NPC1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5218869 0.94 C5AR1 (0.37) C5AR1PTGDR2TSPOGNRHRCNR2
SCHEMBL648586 0.90 C5AR1 (0.39) C5AR1TSPOMAPTRXFP1PPARG
SCHEMBL5633847 0.90 C5AR1 (0.53) C5AR1GNRHRMAPTPPARGPPARA
SCHEMBL5225249 0.89 C5AR1 (0.38) C5AR1PTGDR2GNRHRMAPTCNR2
SCHEMBL648694 0.88 C5AR1 (0.39) C5AR1TSPOGNRHRMAPTRXFP1
SCHEMBL648900 0.86 C5AR1 (0.42) C5AR1MAPTNR1H3PPARGPPARA
SCHEMBL651426 0.85 C5AR1 (0.38) C5AR1PPARGHDAC1PARP1
SCHEMBL648253 0.85 TSHR (0.41) C5AR1TSPOGNRHRMAPTRXFP1
SCHEMBL650278 0.85 C5AR1 (0.40) C5AR1TSPOCNR2PPARGHDAC1
SCHEMBL648873 0.84 MC4R (0.37) C5AR1NR1H3PPARGHDAC1PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7186734-B2 Aryl imidazoles and related compounds as C5a receptor modulators NEUROGEN CORPORATION (US) 2007-03-06 US disclosed