SCHEMBL5634348

SCHEMBL5634348

CCC(C)(CC)OC(=O)NC(Cc1cc(F)c(F)cc1F)C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.43
CTSS P25774 6/20 0.42
CTSK P43235 5/20 0.42
ACE P12821 4/20 0.41
DPP4 P27487 5/20 0.40
SCN9A Q15858 1/20 0.38
ITGB3 P05106 1/20 0.37
ITGA2B P08514 1/20 0.37
MME P08473 2/20 0.37
CPA1 P15085 2/20 0.37
ACE2 Q9BYF1 2/20 0.37
PPARA Q07869 2/20 0.35
PPARG P37231 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5634343 1.00 PTPN1 (0.43) PTPN1CTSSCTSKACEDPP4
SCHEMBL1509374 0.88 PTPN1 (0.53) PTPN1CTSSCTSKACEDPP4
SCHEMBL1509372 0.88 PTPN1 (0.53) PTPN1CTSSCTSKACEDPP4
SCHEMBL30599288 0.88 PTPN1 (0.53) PTPN1CTSSCTSKACEDPP4
SCHEMBL18124300 0.88 PTPN1 (0.53) PTPN1CTSSCTSKACEDPP4
SCHEMBL29398092 0.88 PTPN1 (0.53) PTPN1CTSSCTSKACEDPP4
SCHEMBL29162457 0.80 PTPN1 (0.50) PTPN1CTSSCTSKACESCN9A
SCHEMBL1509413 0.79 PTPN1 (0.49) PTPN1CTSSCTSKACESCN9A
SCHEMBL1509411 0.79 PTPN1 (0.49) PTPN1CTSSCTSKACESCN9A
SCHEMBL16448118 0.78 PTPN1 (0.48) PTPN1CTSSCTSKACESCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7259160-B2 Hexahydrodiazepinones as dipeptidyl peptidase-IV inhibitors for the treatment or prevention of diabetes MERCK & CO., INC. (US) 2007-08-21 US disclosed
US-20060211682-A1 Hexahydrodiazepinones as dipeptidyl peptidase-iv inhibitors for the treatment or prevention of diabetes MERCK SHARP & DOHME LLC 2006-09-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060211682-A1 Hexahydrodiazepinones as dipeptidyl peptidase-iv inhibitors for the treatment or prevention of diabetes DPP4, DPP3, DPP7 PTPN1 1435/4885CTSS 933/4885CTSK 727/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.