SCHEMBL5636052

SCHEMBL5636052

Fc1cccc(-c2cc3c4c(c2)[C@@H]2CNCC[C@@H]2N4CCO3)c1F

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 10/20 0.52
HTR2A P28223 8/20 0.40
HTR2B P41595 3/20 0.40
DRD2 P14416 4/20 0.34
HTR1A P08908 1/20 0.34
DRD4 P21917 1/20 0.34
ADRA1A P35348 1/20 0.34
ADRA1B P35368 1/20 0.34
HTR6 P50406 1/20 0.32
ROCK2 O75116 2/20 0.32
AKT1 P31749 2/20 0.32
PRKCQ Q04759 1/20 0.32
WNT1 P04628 1/20 0.32
DYRK1A Q13627 1/20 0.32
CNR2 P34972 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5637932 0.84 HTR2C (0.43) HTR2CHTR2AHTR2BDRD2HTR1A
SCHEMBL5636741 0.84 HTR2C (0.48) HTR2CHTR2AHTR2BDRD2HTR1A
SCHEMBL5635087 0.84 HTR2C (0.42) HTR2CHTR2AHTR2BDRD2HTR1A
SCHEMBL5638526 0.83 HTR2C (0.44) HTR2CHTR2AHTR2BDRD2ROCK2
SCHEMBL6752904 0.83 HTR2C (0.51) HTR2CHTR2AHTR2B
Hydrochloric Acid SCHEMBL5635163 0.83 HTR2C (0.65) HTR2CHTR2AHTR2BDRD2HTR1A
SCHEMBL5636911 0.83 HTR2C (0.47) HTR2CHTR2AHTR2BDRD2HTR1A
SCHEMBL5636979 0.83 HTR2C (0.46) HTR2CHTR2AHTR2BDRD2HTR1A
SCHEMBL5639194 0.82 HTR2C (0.46) HTR2CHTR2AHTR2BHTR1AHTR6
SCHEMBL5636753 0.82 HTR2C (0.41) HTR2CHTR2AHTR2BDRD2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed