SCHEMBL5636095

SCHEMBL5636095

COCc1cc(OC)ccc1-c1cc2c3c(c1)[C@@H]1CNCC[C@@H]1N3CCCS2

nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 10/20 0.58
HTR2B P41595 6/20 0.54
HTR2A P28223 4/20 0.54
DRD2 P14416 1/20 0.31
ROCK2 O75116 1/20 0.30
KCNH2 Q12809 1/20 0.30
RYR2 Q92736 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5637149 0.92 HTR2C (0.59) HTR2CHTR2BHTR2ADRD2RYR2
SCHEMBL5636799 0.92 HTR2C (0.56) HTR2CHTR2BHTR2A
SCHEMBL6752987 0.92 HTR2C (0.58) HTR2CHTR2BHTR2ADRD2KCNH2
SCHEMBL5636294 0.92 HTR2C (0.58) HTR2CHTR2BHTR2ADRD2
SCHEMBL5636958 0.89 HTR2C (0.62) HTR2CHTR2BHTR2AKCNH2RYR2
SCHEMBL5638466 0.88 HTR2C (0.61) HTR2CHTR2BHTR2AKCNH2RYR2
SCHEMBL5636633 0.87 HTR2C (0.61) HTR2CHTR2BHTR2ADRD2KCNH2
SCHEMBL5636700 0.87 HTR2C (0.68) HTR2CHTR2BHTR2ADRD2
SCHEMBL5636580 0.85 HTR2C (0.58) HTR2CHTR2BHTR2ADRD2RYR2
SCHEMBL5636494 0.85 HTR2C (0.58) HTR2CHTR2BHTR2ADRD2RYR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed