SCHEMBL5636191

SCHEMBL5636191

Clc1ccc(Cl)c(-c2cc3c4c(c2)[C@H]2CNCC[C@H]2N4CCCS3)c1

nearest known ligand 0.66

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 16/20 0.66
HTR2A P28223 13/20 0.59
HTR2B P41595 5/20 0.59
DRD2 P14416 6/20 0.39
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32
KCNH2 Q12809 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5636247 0.92 HTR2C (0.76) HTR2CHTR2AHTR2BDRD2
SCHEMBL255569 0.92 HTR2C (0.76) HTR2CHTR2AHTR2BDRD2
SCHEMBL5637199 0.89 HTR2C (0.69) HTR2CHTR2AHTR2BDRD2
SCHEMBL5637715 0.89 HTR2C (0.64) HTR2CHTR2AHTR2BDRD2
SCHEMBL5637068 0.88 HTR2C (0.70) HTR2CHTR2AHTR2BDRD2
SCHEMBL5636606 0.86 HTR2C (0.63) HTR2CHTR2AHTR2BDRD2KCNH2
Hydrochloric Acid SCHEMBL5637637 0.86 HTR2C (0.67) HTR2CHTR2AHTR2BDRD2
SCHEMBL5635089 0.86 HTR2C (0.73) HTR2CHTR2AHTR2BDRD2
SCHEMBL5636211 0.86 HTR2C (0.70) HTR2CHTR2AHTR2BDRD2
SCHEMBL5637561 0.86 HTR2C (0.70) HTR2CHTR2AHTR2BDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed