SCHEMBL5637101

SCHEMBL5637101

CC(C)(C)OC(=O)N1CCC2C(C1)c1cccc3c1N2CCS3

nearest known ligand 0.50

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 20/20 0.50
HTR2C P28335 20/20 0.50
DRD2 P14416 18/20 0.49
HTR2B P41595 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5637242 0.95 HTR2A (0.54) HTR2AHTR2CDRD2HTR2B
SCHEMBL5637793 0.93 HTR2A (0.46) HTR2AHTR2CDRD2HTR2B
SCHEMBL5635213 0.88 HTR2A (0.53) HTR2AHTR2CDRD2HTR2B
SCHEMBL5636213 0.83 USP30 (0.40) HTR2AHTR2CDRD2
SCHEMBL5637554 0.83 USP30 (0.40) HTR2AHTR2CDRD2
SCHEMBL5637965 0.83 HTR2C (0.54) HTR2AHTR2CDRD2
SCHEMBL5638532 0.81 HTR2C (0.39) HTR2AHTR2CDRD2HTR2B
SCHEMBL5407748 0.80 HTR2A (0.51) HTR2AHTR2CDRD2
SCHEMBL5407746 0.80 HTR2A (0.51) HTR2AHTR2CDRD2
SCHEMBL5637970 0.80 HTR2C (0.48) HTR2AHTR2CDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed