SCHEMBL5637708

SCHEMBL5637708

CC(=O)c1cc(F)ccc1-c1cc2c3c(c1)[C@@H]1CNCC[C@@H]1N3CCCS2

nearest known ligand 0.65

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 18/20 0.65
HTR2A P28223 16/20 0.53
HTR2B P41595 2/20 0.53
DRD2 P14416 14/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5636580 0.88 HTR2C (0.58) HTR2CHTR2AHTR2BDRD2
SCHEMBL5638318 0.88 HTR2C (0.69) HTR2CHTR2AHTR2BDRD2
SCHEMBL5637598 0.86 HTR2C (0.69) HTR2CHTR2AHTR2BDRD2
SCHEMBL5637044 0.86 HTR2C (0.69) HTR2CHTR2AHTR2BDRD2
SCHEMBL5636122 0.85 HTR2C (0.64) HTR2CHTR2AHTR2BDRD2
SCHEMBL5636673 0.84 HTR2C (0.67) HTR2CHTR2AHTR2BDRD2
SCHEMBL5634998 0.83 HTR2C (0.66) HTR2CHTR2AHTR2BDRD2
SCHEMBL6491607 0.83 HTR2C (0.46) HTR2CHTR2AHTR2BDRD2
SCHEMBL5637921 0.83 HTR2C (0.76) HTR2CHTR2AHTR2BDRD2
SCHEMBL5636652 0.83 HTR2C (0.61) HTR2CHTR2AHTR2BDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed