SCHEMBL5653536

SCHEMBL5653536

CCCn1c(=O)c2c(nc(Cc3ccc(S(C)(=O)=O)cc3)n2CCN(CC)CCO)n(CCc2ccc(N)cc2)c1=O

nearest known ligand 0.63

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 3/20 0.63
ADORA2B P29275 12/20 0.40
ADORA2A P29274 7/20 0.40
ADORA3 P0DMS8 5/20 0.39
KMT2A Q03164 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
PTGS2 P35354 1/20 0.37
TSHR P16473 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CYP3A4 P08684 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1332408 0.91 ADORA1 (0.66) ADORA1ADORA2BADORA2AADORA3TSHR
Hydrochloric Acid SCHEMBL1332578 0.90 ADORA1 (0.65) ADORA1ADORA2BADORA2AADORA3TSHR
SCHEMBL1332532 0.90 ADORA1 (0.65) ADORA1ADORA2BADORA2AADORA3KMT2A
SCHEMBL1332766 0.89 ADORA1 (0.63) ADORA1ADORA2BADORA2AADORA3KMT2A
SCHEMBL4176173 0.88 ADORA1 (0.62) ADORA1ADORA2BADORA2AADORA3KMT2A
SCHEMBL1333086 0.88 ADORA1 (0.64) ADORA1ADORA2BADORA2AADORA3KMT2A
SCHEMBL1332444 0.87 ADORA1 (0.62) ADORA1ADORA2BADORA2AADORA3KMT2A
SCHEMBL1334671 0.86 ADORA1 (0.60) ADORA1ADORA2BADORA2AADORA3KMT2A
SCHEMBL1333191 0.86 ADORA1 (0.62) ADORA1ADORA2BADORA2AADORA3TSHR
SCHEMBL1334308 0.86 ADORA1 (0.57) ADORA1ADORA2BADORA2AADORA3TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7247639-B2 A1 adenosine receptor antagonists ENDACEA, INC. (US) 2007-07-24 US claimed