SCHEMBL5658005

SCHEMBL5658005

Cc1cc2c(NC(=O)NCc3ccc(C(F)(F)F)cc3)cccc2c(C)n1

nearest known ligand 0.65

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 13/20 0.65
MAPT P10636 1/20 0.51
KDM4E B2RXH2 2/20 0.48
NAMPT P43490 1/20 0.48
MTOR P42345 1/20 0.48
GSK3B P49841 1/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
ALDH1A1 P00352 1/20 0.47
RAB9A P51151 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4028233 0.90 TRPV1 (0.64) TRPV1MAPTKDM4EGSK3BMEN1
SCHEMBL4023614 0.85 TRPV1 (0.51) TRPV1KDM4EMEN1KMT2AALDH1A1
SCHEMBL4022124 0.85 TRPV1 (0.54) TRPV1KDM4EGSK3BMEN1KMT2A
SCHEMBL4025617 0.85 TRPV1 (0.72) TRPV1
SCHEMBL5659449 0.84 MAPT (0.73) TRPV1MAPTKDM4ENAMPTMTOR
SCHEMBL5658543 0.83 TRPV1 (0.67) TRPV1KDM4ENAMPTMTORGSK3B
SCHEMBL5658216 0.83 TRPV1 (0.72) TRPV1KDM4EGSK3BMEN1KMT2A
SCHEMBL5661327 0.80 TRPV1 (0.61) TRPV1KDM4ENAMPTMTORGSK3B
SCHEMBL5658815 0.80 TRPV1 (0.55) TRPV1MAPTNAMPTMTOR
SCHEMBL12846743 0.78 KMT2A (0.76) TRPV1MAPTNAMPTMTORMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7285563-B2 Heteroaromatic urea derivatives as VR-1 receptor modulators for treating pain MERCK SHARP & DOHME LTD. (GB) 2007-10-23 US disclosed
US-20050107388-A1 Heteroaromatic urea derivatives as vr-1receptor modulators for treating pain MERCK SHARP & DOHME LTD. (GB) 2005-05-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050107388-A1 Heteroaromatic urea derivatives as vr-1receptor modulators for treating pain ARRB1, OPRL1, CNR1 TRPV1 37/4885MAPT 4195/4885KDM4E 3121/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.