SCHEMBL5665269

SCHEMBL5665269

C[Sn](C)(C)c1ccccc1Cl

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.56
LMNA P02545 1/20 0.56
ALDH1A1 P00352 4/20 0.38
CYP2A6 P11509 4/20 0.35
CYP1A2 P05177 3/20 0.35
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33
PNMT P11086 1/20 0.33
IDO1 P14902 1/20 0.33
TAAR1 Q96RJ0 3/20 0.32
HSD11B1 P28845 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8678832 0.78 TSHR (0.35) TSHRLMNACYP2A6CYP1A2
1,2-Dichlorobenzene SCHEMBL28433310 0.75 TSHR (0.83) TSHRLMNAALDH1A1CYP2A6CYP1A2
1,2-Dichlorobenzene SCHEMBL10593125 0.74
1,2-Dichlorobenzene SCHEMBL5190 0.74
1,2-Dichlorobenzene SCHEMBL29350623 0.74
1,2-Dichlorobenzene SCHEMBL1155123 0.74 TSHR (1.00) TSHRLMNAALDH1A1CYP2A6CYP1A2
SCHEMBL23043148 0.74 CYP1A2 (0.38) TSHRLMNAALDH1A1CYP2A6CYP1A2
SCHEMBL29931540 0.74 CYP1A2 (0.38) TSHRLMNAALDH1A1CYP2A6CYP1A2
1,2-Dichlorobenzene SCHEMBL29291037 0.72 TSHR (0.77) TSHRLMNAALDH1A1CYP2A6CYP1A2
1,2-Dichlorobenzene SCHEMBL9662162 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-7038070-B2 Preparation of preparing substituted indanones BASELL POLYOLEFINE GMBH (DE) 2006-05-02 US disclosed
US-6963017-B2 Preparation of preparing substituted indanones BASELL POLYOLEFINE GMBH (DE) 2005-11-08 US disclosed
EP-0968158-B1 METHOD OF PREPARING SUBSTITUTED INDANONES, THE SUBSTITUTED INDANONES AND METALLOCENES PREPARED THEREFROM BASELL POLYOLEFINE GMBH (DE) 2005-08-10 EP disclosed
US-20050033076-A1 Preparation of preparing substituted indanones EQUISTAR CHEMICALS, LP 2005-02-10 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed
US-20030009046-A1 Preparation of preparing substituted indanones EQUISTAR CHEMICALS, LP 2003-01-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050033076-A1 Preparation of preparing substituted indanones CYP1A2, CYP2J2, IDH3A TSHR 4624/4885LMNA 1082/4885ALDH1A1 317/4885
US-20030009046-A1 Preparation of preparing substituted indanones CYP1A2, CYP1B1, CYP1A1 TSHR 4667/4885LMNA 1251/4885ALDH1A1 198/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.