SCHEMBL5670932

SCHEMBL5670932

C=CCN1C(=O)N(c2cccc(C(F)(F)F)c2)C(C)=C(C(=O)O)C1c1ccc(C#N)cc1

nearest known ligand 0.74

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ELANE P08246 20/20 0.74
CYP2C9 P11712 4/20 0.74
CYP3A4 P08684 3/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL395510 1.00 ELANE (0.74) ELANECYP2C9CYP3A4
SCHEMBL1245162 0.95 ELANE (0.79) ELANECYP2C9CYP3A4
SCHEMBL1764354 0.90 ELANE (0.77) ELANECYP2C9CYP3A4
SCHEMBL13872750 0.90 ELANE (0.77) ELANECYP2C9CYP3A4
SCHEMBL3482734 0.90 ELANE (0.77) ELANECYP2C9CYP3A4
SCHEMBL14899953 0.89 ELANE (0.90) ELANECYP2C9CYP3A4
SCHEMBL6025373 0.88 ELANE (0.74) ELANECYP2C9CYP3A4
SCHEMBL394959 0.88 ELANE (0.74) ELANECYP2C9CYP3A4
SCHEMBL1155480 0.87 ELANE (0.63) ELANECYP2C9
SCHEMBL4317225 0.87 ELANE (0.82) ELANECYP2C9CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730121-A2 1,4-DIARYL-DIHYDROPYRIMIDIN-2-ONES AND THEIR USE AS HUMAN NEUTROPHIL ELASTASE INHIBITORS Bayer HealthCare AG (DE) 2006-12-13 EP disclosed
WO-2005082863-A2 1,4 DIARYL-DIHYDROPYRIMIDIN-2 ONES AND THEIR USE AS A HUMAN NEUTROPHIL ELASTASE INHIBITORS BAYER HEALTHCARE AG (DE) 2005-09-09 WO disclosed