SCHEMBL5675600

SCHEMBL5675600

CCC/C=C/S(=O)(=O)NC(=O)/C=C/c1c(Cl)nc(C)n1Cc1ccc(NC(=O)OC(C)(C)C)cc1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 5/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36
ALDH1A1 P00352 2/20 0.34
MAPT P10636 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
RORC P51449 2/20 0.34
KDM4E B2RXH2 1/20 0.34
HPGD P15428 1/20 0.34
HTT P42858 1/20 0.34
HSD17B10 Q99714 1/20 0.34
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
AGTR1 P30556 3/20 0.33
AGTR2 P50052 3/20 0.33
PTGER3 P43115 2/20 0.33
ACSS2 Q9NR19 1/20 0.33
MAPKAPK2 P49137 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5675605 1.00 PPARG (0.36) PPARGPTGDR2ALDH1A1MAPTSMN1; SMN2
SCHEMBL5675418 0.90 PTGDR2 (0.43) PTGDR2ALDH1A1MAPTSMN1; SMN2RORC
SCHEMBL5675423 0.90 PTGDR2 (0.43) PTGDR2ALDH1A1MAPTSMN1; SMN2RORC
SCHEMBL5675542 0.88 PPARG (0.48) PPARGPTGDR2
SCHEMBL5675551 0.88 PPARG (0.48) PPARGPTGDR2
SCHEMBL5673981 0.85 PTGDR2 (0.40) PTGDR2ALDH1A1MAPTSMN1; SMN2RORC
SCHEMBL5673971 0.85 PTGDR2 (0.40) PTGDR2ALDH1A1MAPTSMN1; SMN2RORC
SCHEMBL5213112 0.82 PPARG (0.42) PPARGHDAC8
SCHEMBL5213109 0.82 PPARG (0.42) PPARGHDAC8
SCHEMBL5675452 0.82 HDAC1 (0.41) PPARGPTGDR2ALDH1A1MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1142879-A1 IMIDAZOLE COMPOUNDS AND MEDICINAL USE THEREOF FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-10-10 EP claimed
US-7060721-B1 Imidazole compounds and medicinal use thereof FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2006-06-13 US disclosed
EP-1142879-A1 IMIDAZOLE COMPOUNDS AND MEDICINAL USE THEREOF FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-10-10 EP disclosed