SCHEMBL5684294

SCHEMBL5684294

CCCC1CCc2c(ccc3c2CCC(CCc2cc(F)c(OC(F)(F)F)c(F)c2)C3)C1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 6/20 0.36
DRD2 P14416 5/20 0.36
CYP3A4 P08684 1/20 0.34
CYP2C8 P10632 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
S1PR3 Q99500 1/20 0.34
HTR1D P28221 1/20 0.32
HTR1B P28222 1/20 0.32
CYP19A1 P11511 1/20 0.31
HCRTR1 O43613 2/20 0.31
HCRTR2 O43614 2/20 0.31
FYN P06241 1/20 0.31
CHRM2 P08172 1/20 0.30
CHRM5 P08912 1/20 0.30
CHRM1 P11229 1/20 0.30
CHRM3 P20309 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5684987 0.87 HCRTR1 (0.39) DRD3DRD2CYP3A4CYP2C8CYP2D6
SCHEMBL5683897 0.86 HTR1D (0.32) DRD3DRD2CYP3A4CYP2C8S1PR3
SCHEMBL5684743 0.85 HTR1D (0.36) DRD3DRD2CYP3A4CYP2C8CYP2D6
SCHEMBL5686395 0.85 HTR1D (0.36) DRD3DRD2CYP3A4CYP2C8CYP2D6
SCHEMBL8747891 0.83 CHRM2 (0.32) CHRM2CHRM5CHRM1CHRM3
SCHEMBL5683468 0.83 SLC6A4 (0.40) DRD3DRD2CYP3A4CYP2C8CYP2D6
SCHEMBL5684977 0.82 HTR1D (0.35) DRD3DRD2CYP3A4CYP2C8CYP2D6
SCHEMBL5685005 0.81 CYP3A4 (0.39) DRD3DRD2CYP3A4CYP2C8CYP2D6
SCHEMBL5684416 0.81 CYP3A4 (0.39) DRD3DRD2CYP3A4CYP2C8CYP2D6
SCHEMBL8095326 0.81 CHRM2 (0.32) CHRM2CHRM5CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7067179-B1 Fused ring compound DAINIPPON INK AND CHEMICALS, INC. (JP) 2006-06-27 US disclosed
EP-1201632-B1 FUSED RING COMPOUND DAINIPPON INK & CHEMICALS (JP) 2006-03-29 EP disclosed
EP-1201632-A1 FUSED RING COMPOUND DAINIPPON INK AND CHEMICALS, INC. (JP) 2002-05-02 EP disclosed