SCHEMBL5688690

SCHEMBL5688690

CC(C)C(O)(c1cccc(-c2ccccn2)c1)c1c[nH]cn1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 11/20 0.51
CYP3A4 P08684 10/20 0.51
HRH3 Q9Y5N1 1/20 0.36
TGFBR1 P36897 1/20 0.36
HTR1A P08908 1/20 0.35
HTR7 P34969 1/20 0.35
CNR1 P21554 1/20 0.35
KAT6A Q92794 1/20 0.34
CTSL P07711 1/20 0.34
CTSK P43235 1/20 0.34
AXL P30530 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18770487 0.87 CYP17A1 (0.63) CYP17A1CYP3A4
SCHEMBL5690534 0.87 CYP17A1 (0.60) CYP17A1CYP3A4
SCHEMBL5688702 0.83 CYP17A1 (0.53) CYP17A1CYP3A4
SCHEMBL5688302 0.81 CYP17A1 (0.46) CYP17A1CYP3A4HTR1AHTR7CNR1
SCHEMBL5688560 0.81 CYP3A4 (0.51) CYP17A1CYP3A4AXL
SCHEMBL5688934 0.81 CYP17A1 (0.52) CYP17A1CYP3A4
SCHEMBL5688356 0.81 CYP17A1 (0.50) CYP17A1CYP3A4
SCHEMBL5691318 0.80 CYP17A1 (0.58) CYP17A1CYP3A4
SCHEMBL5691340 0.80 CYP17A1 (0.63) CYP17A1CYP3A4CNR1
SCHEMBL5688515 0.80 CYP17A1 (0.63) CYP17A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1227086-B1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2006-03-29 EP disclosed
US-6518257-B1 1-substituted phenyl-1-(1h-imidazol-4-yl) alcohols, process for producing the same and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-02-11 US disclosed
EP-1227086-A1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-07-31 EP disclosed