SCHEMBL5689337

SCHEMBL5689337

CN(CCCc1ccc(F)cc1)[C@H]1CC[C@H](c2ccc(O)cc2)CC1

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SPHK1 Q9NYA1 2/20 0.49
AGTR2 P50052 3/20 0.42
KDM4E B2RXH2 1/20 0.41
ESR2 Q92731 1/20 0.41
KCNH2 Q12809 1/20 0.41
GRIN2B Q13224 1/20 0.41
ALOX5 P09917 1/20 0.40
CHIT1 Q13231 1/20 0.40
CHIA Q9BZP6 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5689334 1.00 SPHK1 (0.49) SPHK1AGTR2KDM4EESR2KCNH2
SCHEMBL5689661 0.87 KDM4E (0.52) SPHK1KDM4EGRIN2B
SCHEMBL6841392 0.87 KDM4E (0.56) SPHK1KDM4EGRIN2B
SCHEMBL5689666 0.87 KDM4E (0.52) SPHK1KDM4EGRIN2B
SCHEMBL6836225 0.87 KDM4E (0.56) SPHK1KDM4EGRIN2B
SCHEMBL7023319 0.87 KDM4E (0.52) SPHK1KDM4EGRIN2B
SCHEMBL6840856 0.84 KDM4E (0.54) SPHK1KDM4EGRIN2B
SCHEMBL6840853 0.84 KDM4E (0.54) SPHK1KDM4EGRIN2B
SCHEMBL5690171 0.82 BCHE (0.47) SPHK1KDM4EGRIN2BALOX5
SCHEMBL5690175 0.82 BCHE (0.47) SPHK1KDM4EGRIN2BALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0982026-B1 Use of aryl-cyclohexylamine derivatives in the manufacture of NMDA receptor blockers HOFFMANN LA ROCHE (CH) 2006-05-17 EP claimed
US-6184236-B1 Method of treating a neurodegenerative disease by administering an aryl-cyclohexylamine derivative HOFFMANN-LA ROCHE INC. 2001-02-06 US claimed
EP-0982026-A2 Use of aryl-cyclohexylamine derivatives in the manufacture of NMDA receptor blockers F. HOFFMANN-LA ROCHE AG (CH) 2000-03-01 EP claimed
EP-0982026-B1 Use of aryl-cyclohexylamine derivatives in the manufacture of NMDA receptor blockers HOFFMANN LA ROCHE (CH) 2006-05-17 EP disclosed
US-6184236-B1 Method of treating a neurodegenerative disease by administering an aryl-cyclohexylamine derivative HOFFMANN-LA ROCHE INC. 2001-02-06 US disclosed
EP-0982026-A2 Use of aryl-cyclohexylamine derivatives in the manufacture of NMDA receptor blockers F. HOFFMANN-LA ROCHE AG (CH) 2000-03-01 EP disclosed