SCHEMBL5693752

SCHEMBL5693752

CC(=Nc1c(C)cc(C)cc1C)c1cccc(C(C)=Nc2c(C)cc(C)cc2C)n1.CC(=Nc1c(C)cc(C)cc1C)c1cccc(C(C)=Nc2c(C)cc(C)cc2C)n1.[Co+].[Co+].[O-]c1c([O-])c2ccccc2c2ccccc12

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.35
CYP2A6 P11509 1/20 0.35
PAX8 Q06710 1/20 0.34
NPFFR1 Q9GZQ6 1/20 0.33
NPFFR2 Q9Y5X5 1/20 0.33
HDAC6 Q9UBN7 1/20 0.32
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
NPC1 O15118 1/20 0.31
MAPT P10636 1/20 0.31
RAB9A P51151 1/20 0.31
ALDH1A1 P00352 2/20 0.31
THRB P10828 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5693796 0.91 HDAC6 (0.36) CYP1A2CYP2A6PAX8NPFFR1NPFFR2
SCHEMBL453478 0.86 HSP90AA1 (0.36) CYP1A2CYP2A6PAX8NPFFR1NPFFR2
SCHEMBL453477 0.86 HSP90AA1 (0.36) CYP1A2CYP2A6PAX8NPFFR1NPFFR2
SCHEMBL5693842 0.85 CYP1A2 (0.33) CYP1A2CYP2A6PAX8ALDH1A1
SCHEMBL5693760 0.85 MAPT (0.47) CYP1A2PAX8HDAC6MEN1KMT2A
SCHEMBL5588611 0.84 HSP90AA1 (0.35) CYP1A2CYP2A6PAX8NPFFR1NPFFR2
SCHEMBL5588127 0.84 HSP90AA1 (0.35) CYP1A2CYP2A6PAX8NPFFR1NPFFR2
SCHEMBL5587833 0.84 HSP90AA1 (0.35) CYP1A2CYP2A6PAX8NPFFR1NPFFR2
SCHEMBL5588774 0.84 HSP90AA1 (0.35) CYP1A2CYP2A6PAX8NPFFR1NPFFR2
SCHEMBL5587427 0.84 HSP90AA1 (0.35) CYP1A2CYP2A6PAX8NPFFR1NPFFR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1521758-B1 LATE TRANSITION METAL CATALYSTS FOR OLEFIN POLYMERIZATION AND OLIGOMERIZATION EXXONMOBIL CHEM PATENTS INC (US) 2006-05-24 EP claimed