SCHEMBL5696608

SCHEMBL5696608

O=C(CO)N1CCCCC1COc1cccc2ncnc(Nc3ccc(O)c(Cl)c3)c12

nearest known ligand 0.73

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 17/20 0.73
EGFR P00533 13/20 0.73
KCNH2 Q12809 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4389877 1.00 ERBB2 (0.73) ERBB2EGFRKCNH2
SCHEMBL4390846 1.00 ERBB2 (0.73) ERBB2EGFRKCNH2
SCHEMBL4390515 0.98 ERBB2 (0.76) ERBB2EGFRKCNH2
SCHEMBL4383257 0.98 ERBB2 (0.76) ERBB2EGFRKCNH2
SCHEMBL5696689 0.98 ERBB2 (0.76) ERBB2EGFRKCNH2
SCHEMBL4389102 0.91 ERBB2 (0.61) ERBB2EGFRKCNH2
SCHEMBL5696875 0.91 ERBB2 (0.64) ERBB2EGFRKCNH2
SCHEMBL4396280 0.91 ERBB2 (0.64) ERBB2EGFRKCNH2
SCHEMBL5696654 0.88 ERBB2 (0.64) ERBB2EGFRKCNH2
SCHEMBL4395376 0.88 ERBB2 (0.64) ERBB2EGFRKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1664029-A1 QUINAZOLINE DERIVATIVES AS ANTITUMOR AGENTS AstraZeneca AB (SE) 2006-06-07 EP disclosed
WO-2005026152-A1 QUINAZOLINE DERIVATIVES AS ANTITUMOR AGENTS ASTRAZENECA AB (SE) 2005-03-24 WO disclosed