SCHEMBL5711276

SCHEMBL5711276

O=CCC[C@H]1C(=O)OCN1C(=O)OCc1ccccc1

nearest known ligand 0.64

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.64
PSEN1 P49768 1/20 0.46
PSEN2 P49810 1/20 0.46
APH1B Q8WW43 1/20 0.46
NCSTN Q92542 1/20 0.46
APH1A Q96BI3 1/20 0.46
PSENEN Q9NZ42 1/20 0.46
ELANE P08246 3/20 0.44
F2 P00734 2/20 0.44
CTSG P08311 1/20 0.44
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5711245 1.00 USP2 (0.64) USP2PSEN1PSEN2APH1BNCSTN
SCHEMBL8694697 1.00 USP2 (0.64) USP2PSEN1PSEN2APH1BNCSTN
SCHEMBL5711344 0.93 USP2 (0.61) USP2PSEN1PSEN2APH1BNCSTN
SCHEMBL5711222 0.93 USP2 (0.61) USP2PSEN1PSEN2APH1BNCSTN
SCHEMBL5711223 0.92 USP2 (0.60) USP2PSEN1PSEN2APH1BNCSTN
SCHEMBL5711372 0.88 USP2 (0.66) USP2PSEN1PSEN2APH1BNCSTN
SCHEMBL6965437 0.87 USP2 (0.64) USP2PSEN1PSEN2APH1BNCSTN
SCHEMBL3184957 0.86 USP2 (0.63) USP2PSEN1PSEN2APH1BNCSTN
SCHEMBL5711299 0.86 USP2 (0.63) USP2PSEN1PSEN2APH1BNCSTN
SCHEMBL8842431 0.86 USP2 (0.63) USP2PSEN1PSEN2APH1BNCSTN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230151060-A1 CYCLIC PEPTIDE COMPOUND HAVING KRAS INHIBITORY ACTION CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2023-05-18 US disclosed
US-20230151060-A1 CYCLIC PEPTIDE COMPOUND HAVING KRAS INHIBITORY ACTION CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2023-05-18 US disclosed
WO-2022234853-A1 CYCLIC COMPOUND HAVING INHIBITORY EFFECT SELECTIVE FOR KRAS BUT NOT FOR HRAS AND NRAS 中外製薬株式会社 2022-11-10 WO disclosed
US-20100280120-A1 COMPOUND INDUCING ANGIOGENESIS RESPONSE IN ISCHAEMIC TISSUES Green Cross Therapeutics Private Limited (IN) 2010-11-04 US disclosed
EP-1103560-B1 NOVEL THIAZOLIDINE DERIVATIVES SANTEN PHARMACEUTICAL CO LTD (JP) 2006-12-27 EP disclosed
EP-1103560-A1 NOVEL THIAZOLIDINE DERIVATIVES SANTEN PHARMACEUTICAL CO., LTD. (JP) 2001-05-30 EP disclosed
US-5710129-A Inhibitors of SH2-mediated processes ARIAD PHARMACEUTICALS, INC. (US) 1998-01-20 US disclosed
WO-1997031016-A2 NEW INHIBITORS OF SH2-MEDIATED PROCESSES ARIAD PHARMACEUTICALS, INC. (US) 1997-08-28 WO disclosed
US-5658945-A ANTICANCER AGENT; AIDS THERAPY; CONTROLLING INFECTIONS AMERICAN CYANAMID COMPANY (US) 1997-08-19 US disclosed
US-5633280-A ACCELERATED RECOVERY FROM CHEMOTHERAPY, RADIATION TREATMENT, BONE MARROW TRANSPLANTATION, INFECTIONS AMERICAN CYANAMID COMPANY (US) 1997-05-27 US disclosed
US-5616612-A THERAPY FOR CANCER, AIDS, ANEMIA, INFECTIONS AMERICAN CYANAMID COMPANY (US) 1997-04-01 US disclosed
US-5602275-A MAY BE USED TO ACCELERATE RECOVERY FROM NEUTROPENIA ACCOMPANYING RADIO- OR CHEMOTHERAPY, BONE MARROW TRANSPLANTATION OR INFECTIONS AMERICAN CYANAMID COMPANY (US) 1997-02-11 US disclosed
EP-0652228-B1 Urethanes and ureas that induce cytokine production AMERICAN CYANAMID CO (US) 1996-10-23 EP disclosed
US-5545662-A USED TO ACCELERATE RECOVERY FROM NEUTROPENIA ACCOMPANYING RADIO OR CHEMOTHERAPY, BONE MARROW TRANSPLANTATION, OR INFECTIONS AMERICAN CYANAMID COMPANY (US) 1996-08-13 US disclosed
EP-0652228-A1 Urethanes and ureas that induce cytokine production AMERICAN CYANAMID COMPANY (US) 1995-05-10 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230151060-A1 CYCLIC PEPTIDE COMPOUND HAVING KRAS INHIBITORY ACTION KRAS, NRAS, HRAS USP2 2527/4885PSEN1 3502/4885PSEN2 3673/4885
US-20100280120-A1 COMPOUND INDUCING ANGIOGENESIS RESPONSE IN ISCHAEMIC TISSUES FLT4, TEK, VEGFA USP2 4602/4885PSEN1 4783/4885PSEN2 4758/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.