SCHEMBL5712903

SCHEMBL5712903

N[C@H]1COc2ccccc2N(CC(=O)OCc2ccccc2)C1=O

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MME P08473 3/20 0.48
ACE P12821 3/20 0.48
P2RX1 P51575 1/20 0.43
P2RX3 P56373 1/20 0.43
P2RX4 Q99571 1/20 0.43
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
TSHR P16473 1/20 0.41
AVPR1A P37288 1/20 0.41
CCKBR P32239 1/20 0.40
ALDH1A1 P00352 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
HPGD P15428 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
RIPK1 Q13546 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7283214 1.00 MME (0.48) MMEACEP2RX1P2RX3P2RX4
Hydrochloric Acid SCHEMBL5712964 0.99 MME (0.48) MMEACEP2RX1P2RX3P2RX4
Hydrochloric Acid SCHEMBL7279438 0.99 MME (0.48) MMEACEP2RX1P2RX3P2RX4
SCHEMBL2687108 0.83 MME (0.55) MMEACENPC1RAB9AALDH1A1
SCHEMBL200386 0.83 MME (0.55) MMEACENPC1RAB9AALDH1A1
SCHEMBL200387 0.83 MME (0.55) MMEACENPC1RAB9AALDH1A1
SCHEMBL7290163 0.81 MAPT (0.43) CCKBRSMN1; SMN2
SCHEMBL7290156 0.81 MAPT (0.43) CCKBRSMN1; SMN2
SCHEMBL17653866 0.80 KMT2A (0.57) TSHRALDH1A1LMNATP53
SCHEMBL7298515 0.79 MME (0.51) MMEACETSHRRIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0135349-B1 CONDENSED SEVEN-MEMBERED RING COMPOUNDS AND THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1988-11-02 EP claimed
EP-0135349-A1 Condensed seven-membered ring compounds and their production and use Takeda Chemical Industries, Ltd. (JP) 1985-03-27 EP claimed
EP-0942925-B1 INHIBITORS OF INTERLEUKIN-1 BETA CONVERTING ENZYME VERTEX PHARMA (US) 2006-11-22 EP disclosed
EP-1466921-A1 Inhibitors of interleukin-1 beta converting enzyme Vertex Pharmaceuticals Incorporated (US) 2004-10-13 EP disclosed
US-6350741-B1 1-BENZAZEPINE DERIVATIVES; ANTIINFLAMMATORY, ANTIARTHRITIC AGENTS; BONE AND AUTOIMMUNE DISORDER TREATMENT VERTEX PHARMACEUTICAL, INC. 2002-02-26 US disclosed